SCHEMBL8868604

SCHEMBL8868604

O=C(O)C(CCCCBr)CCc1cccc2ccccc12

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTNNB1 P35222 1/20 0.46
TDP1 Q9NUW8 1/20 0.45
MTNR1A P48039 2/20 0.43
MCL1 Q07820 4/20 0.41
KMT2A Q03164 1/20 0.41
SLC1A3 P43003 1/20 0.41
SLC1A2 P43004 1/20 0.41
SLC1A1 P43005 1/20 0.41
FOLH1 Q04609 1/20 0.41
CYP1A2 P05177 2/20 0.40
HRH4 Q9H3N8 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8890206 0.89 TDP1 (0.56) CTNNB1TDP1MTNR1AMCL1KMT2A
SCHEMBL1858161 0.83 KMT2A (0.52) CTNNB1TDP1MTNR1AMCL1KMT2A
SCHEMBL8868645 0.80 GRIK1 (0.51) FOLH1CYP1A2
SCHEMBL8867961 0.80 GRIK1 (0.51) FOLH1CYP1A2
SCHEMBL8867562 0.80 GRIK1 (0.51) FOLH1CYP1A2
SCHEMBL1862472 0.78 KMT2A (0.47) TDP1MTNR1AMCL1KMT2A
SCHEMBL10521472 0.76 SIGMAR1 (0.52) CTNNB1TDP1KMT2AFOLH1HRH4
SCHEMBL6680287 0.76 CYP1A2 (0.48) TDP1MTNR1AMCL1CYP1A2CYP2C19
SCHEMBL8868315 0.75 GRIK1 (0.56) TDP1FOLH1CYP1A2
SCHEMBL27584168 0.75 TDP1 (0.54) CTNNB1TDP1MTNR1AMCL1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5599966-A SUITABLE FOR TREATMENT OF DISEASES OF RESPIRATORY PASSAGES BYK NEDERLAND BV (NL) 1997-02-04 US disclosed
WO-1994008945-A1 SUBSTITUTED ETHANOLAMINE ESTERS BYK NEDERLAND BV (NL) 1994-04-28 WO disclosed