SCHEMBL8869757

SCHEMBL8869757

COCCNC(=O)c1ccc(C(=O)NS(=O)(=O)c2ccc(CCNC(=O)c3ccc(OC)c(OC)c3)cc2)cn1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.60
NPC1 O15118 1/20 0.53
RAB9A P51151 1/20 0.53
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
CA7 P43166 1/20 0.52
CA9 Q16790 1/20 0.52
CA14 Q9ULX7 1/20 0.52
ALDH1A1 P00352 3/20 0.50
TP53 P04637 1/20 0.50
MAPT P10636 1/20 0.50
CNR2 P34972 2/20 0.49
NLRP3 Q96P20 2/20 0.49
KMT2A Q03164 2/20 0.48
P4HTM Q9NXG6 1/20 0.48
GAA P10253 1/20 0.48
NAMPT P43490 1/20 0.48
USP2 O75604 1/20 0.48
MAPK1 P28482 1/20 0.48
MEN1 O00255 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8868879 0.95 CA1 (0.60) TSHRCA1CA2CA7CA9
SCHEMBL8868857 0.94 TSHR (0.61) TSHRNPC1RAB9ACA1CA2
SCHEMBL8868796 0.93 TSHR (0.56) TSHRNPC1RAB9ACA1CA2
SCHEMBL8867517 0.93 TSHR (0.56) TSHRNPC1RAB9ACA1CA2
SCHEMBL8868124 0.91 TSHR (0.58) TSHRNPC1RAB9ACA1CA2
SCHEMBL8868966 0.91 TSHR (0.58) TSHRNPC1RAB9ACA1CA2
SCHEMBL8869792 0.91 ALDH1A1 (0.58) TSHRCA1CA2CA7CA9
SCHEMBL8868897 0.90 ALDH1A1 (0.56) TSHRNPC1RAB9ACA1CA2
SCHEMBL7869461 0.89 TSHR (0.57) TSHRNPC1RAB9ACA1CA2
SCHEMBL8868956 0.89 TSHR (0.53) TSHRNPC1RAB9ACA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607954-A Sulfonamido- and sulfonamidocarbonylpyridine-2-carboxamides and their pyridine-n-oxides, process for their preparation and their use as pharmaceuticals HOECHST AKTIENGESELLSCHAFT (DE) 1997-03-04 US disclosed