SCHEMBL8870189

SCHEMBL8870189

c1c2c(cc3c1OCO3)C1Cc3cc4c(cc3C(C2)N1)OCO4

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.53
CYP3A4 P08684 1/20 0.53
DRD1 P21728 2/20 0.42
ADRA1A P35348 1/20 0.42
DRD2 P14416 1/20 0.42
KDM4E B2RXH2 3/20 0.40
ALDH1A1 P00352 2/20 0.40
GLA P06280 2/20 0.40
HPGD P15428 2/20 0.40
CASP1 P29466 2/20 0.40
CASP7 P55210 2/20 0.40
HSD17B10 Q99714 2/20 0.40
CYP2D6 P10635 1/20 0.40
ACHE P22303 1/20 0.40
GAA P10253 1/20 0.39
CHRNA7 P36544 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7999291 1.00 HTR1A (0.53) HTR1ACYP3A4DRD1ADRA1ADRD2
Hydrochloric Acid SCHEMBL8871565 0.98 CYP3A4 (0.51) HTR1ACYP3A4DRD1ADRA1ADRD2
SCHEMBL14883442 0.79 HTR1A (0.49) HTR1ACYP3A4DRD1DRD2
SCHEMBL29866247 0.77 CYP3A4 (0.40) HTR1ACYP3A4DRD1ADRA1ADRD2
SCHEMBL29877224 0.73 CHRNA7 (0.41) HTR1ACYP3A4KDM4EALDH1A1GLA
SCHEMBL6981317 0.69 HTR1A (0.50) HTR1ACYP3A4DRD1ADRA1ADRD2
SCHEMBL7485380 0.69 HTR1A (0.50) HTR1ACYP3A4DRD1ADRA1ADRD2
SCHEMBL3144482 0.69 HTR1A (0.50) HTR1ACYP3A4DRD1ADRA1ADRD2
Escholtzine SCHEMBL29692675 0.69 HTR1A (1.00) HTR1ACYP3A4DRD1ADRA1ADRD2
SCHEMBL9311203 0.69 HTR1A (0.50) HTR1ACYP3A4DRD1ADRA1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5648359-A ESCHSCHOLTZINE AND DERIVATIVES SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1997-07-15 US disclosed
EP-0663210-A2 Tumor necrosis factor production inhibitors SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1995-07-19 EP disclosed