SCHEMBL8870871

SCHEMBL8870871

O=C1c2ccccc2C(=O)N1CCCCN1C2Cc3cc4c(cc3C1Cc1cc3c(cc12)OCO3)OCO4

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.49
CYP3A4 P08684 1/20 0.49
KMT2A Q03164 3/20 0.46
TSHR P16473 2/20 0.46
PKM P14618 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
HSD17B10 Q99714 1/20 0.43
ALDH1A1 P00352 2/20 0.43
USP2 O75604 1/20 0.43
HPGD P15428 1/20 0.43
MAPT P10636 1/20 0.41
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
LMNA P02545 1/20 0.40
DRD3 P35462 2/20 0.40
HTR7 P34969 1/20 0.40
SCN9A Q15858 1/20 0.40
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
SIGMAR1 Q99720 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8871833 0.93 HTR1A (0.51) HTR1ACYP3A4KMT2ATSHRPKM
SCHEMBL8870963 0.77 HTR1A (0.59) HTR1ACYP3A4HSD17B10ALDH1A1HPGD
SCHEMBL9275178 0.76 HTR1A (0.60) HTR1ACYP3A4HSD17B10ALDH1A1HPGD
SCHEMBL8871066 0.73 HTR1A (0.64) HTR1ACYP3A4HSD17B10ALDH1A1HPGD
SCHEMBL8424220 0.71 KMT2A (0.67) KMT2ATSHRPKMSMN1; SMN2HSD17B10
Hydrochloric Acid SCHEMBL8870351 0.71 HTR1A (0.53) HTR1ACYP3A4SIGMAR1DRD2
SCHEMBL8871523 0.70 HTR1A (0.59) HTR1ACYP3A4HSD17B10ALDH1A1HPGD
SCHEMBL8870113 0.70 HTR1A (0.63) HTR1ACYP3A4KMT2AHSD17B10ALDH1A1
SCHEMBL281993 0.69 SCN9A (0.56) HTR1ACYP3A4KMT2ATSHRPKM
Hydrochloric Acid SCHEMBL8871647 0.69 HTR1A (0.66) HTR1ACYP3A4HSD17B10ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5648359-A ESCHSCHOLTZINE AND DERIVATIVES SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1997-07-15 US disclosed
EP-0663210-A2 Tumor necrosis factor production inhibitors SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1995-07-19 EP disclosed