SCHEMBL8872152

SCHEMBL8872152

O=C(O)CN1C(=O)C(=O)N(Cc2cccnc2)C1=O

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.55
NAPRT Q6XQN6 1/20 0.51
KDM4E B2RXH2 1/20 0.50
UBE2N P61088 1/20 0.50
ATM Q13315 1/20 0.50
MAPT P10636 3/20 0.48
RAB9A P51151 1/20 0.47
LMNA P02545 2/20 0.47
ALDH1A1 P00352 2/20 0.46
MEN1 O00255 1/20 0.46
TP53 P04637 1/20 0.46
GAA P10253 1/20 0.46
THRB P10828 1/20 0.46
ALOX15 P16050 1/20 0.46
MAPK1 P28482 1/20 0.46
HTT P42858 1/20 0.46
RECQL P46063 1/20 0.46
HSD17B10 Q99714 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
NLRP3 Q96P20 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8143584 0.83 KMT2A (0.76) KMT2AMAPTRAB9AALDH1A1
SCHEMBL8871897 0.82 KMT2A (0.56) KMT2AMAPTRAB9AALDH1A1
SCHEMBL8873587 0.82 KMT2A (0.67) KMT2AATMALDH1A1MEN1MAPK1
SCHEMBL8136035 0.74 KMT2A (0.78) KMT2AATMMAPT
SCHEMBL8872785 0.74 KMT2A (0.63) KMT2AATMMAPTALDH1A1MEN1
SCHEMBL8144324 0.74 KMT2A (0.58) KMT2AMAPTRAB9AALDH1A1
SCHEMBL8150342 0.73 MAPT (0.68) KMT2AMAPTRAB9ALMNAALDH1A1
SCHEMBL8149456 0.73 KMT2A (0.56) KMT2AMAPTRAB9ALMNAALDH1A1
SCHEMBL8144325 0.73 KMT2A (0.56) KMT2AMAPTRAB9AALDH1A1
SCHEMBL8873707 0.72 ALDH1A1 (0.56) KMT2AKDM4ELMNAALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5681843-A ANTIDIABETIC; ALDOSE REDUCTASE INHIBITOR WITHOUT SUBSTANTIALLY INHIBITING ALDEHYDE REDUCATASE NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 1997-10-28 US disclosed
EP-0718289-A1 Novel parabanic acid derivatives as aldose reductase inhibitors NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 1996-06-26 EP disclosed