SCHEMBL8873641

SCHEMBL8873641

CCOC(=O)CN1C(=O)C(=O)N(Cc2cccc(C(=O)OC)c2)C1=O

nearest known ligand 0.73

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.73
MEN1 O00255 1/20 0.53
ATM Q13315 1/20 0.53
TRPA1 O75762 1/20 0.48
ABHD6 Q9BV23 1/20 0.48
PTPN1 P18031 2/20 0.48
MAPT P10636 3/20 0.48
POLB P06746 2/20 0.48
GAA P10253 1/20 0.48
LOXL2 Q9Y4K0 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8872167 0.89 PTPN1 (0.58) KMT2ATRPA1ABHD6PTPN1MAPT
SCHEMBL8872446 0.87 KMT2A (0.74) KMT2AMEN1ATMPTPN1MAPT
SCHEMBL8871718 0.86 MAPT (0.53) KMT2ATRPA1ABHD6MAPTPOLB
SCHEMBL9322607 0.84 KMT2A (0.76) KMT2AMEN1ATMPTPN1MAPT
SCHEMBL9322643 0.82 KMT2A (0.78) KMT2AMEN1ATMPTPN1MAPT
SCHEMBL9323818 0.81 KMT2A (0.76) KMT2AMEN1ATMPTPN1MAPT
SCHEMBL9322747 0.81 KMT2A (0.71) KMT2AMEN1ATMPTPN1POLB
SCHEMBL8871853 0.80 KMT2A (0.73) KMT2AMEN1ATMPTPN1MAPT
SCHEMBL9325709 0.78 KMT2A (0.67) KMT2AMEN1ATMMAPT
SCHEMBL6978776 0.78 KMT2A (0.70) KMT2AMEN1ATMPTPN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5681843-A ANTIDIABETIC; ALDOSE REDUCTASE INHIBITOR WITHOUT SUBSTANTIALLY INHIBITING ALDEHYDE REDUCATASE NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 1997-10-28 US disclosed
EP-0718289-A1 Novel parabanic acid derivatives as aldose reductase inhibitors NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 1996-06-26 EP disclosed