SCHEMBL8875016

SCHEMBL8875016

CC(=O)OC[C@@H](CCc1ccc(Br)cc1)CO[Si](C)(C)C(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.33
HSP90AA1 P07900 1/20 0.33
POLB P06746 1/20 0.32
CTDSP1 Q9GZU7 1/20 0.32
PPARD Q03181 2/20 0.31
PPARA Q07869 2/20 0.31
MME P08473 1/20 0.31
MMP2 P08253 1/20 0.31
MMP3 P08254 1/20 0.31
KDM4E B2RXH2 3/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
TSHR P16473 1/20 0.31
CYP2C19 P33261 1/20 0.31
MAOB P27338 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
ADRA1A P35348 1/20 0.31
HSD17B10 Q99714 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8875013 1.00 KMT2A (0.33) KMT2AHSP90AA1POLBCTDSP1PPARD
SCHEMBL8875020 1.00 KMT2A (0.33) KMT2AHSP90AA1POLBCTDSP1PPARD
SCHEMBL6506348 0.86 KMT2A (0.40) KMT2AHSP90AA1POLBCTDSP1KDM4E
SCHEMBL8875295 0.84 APP (0.36) KMT2AHSP90AA1
SCHEMBL8875302 0.84 APP (0.36) KMT2AHSP90AA1
SCHEMBL8876633 0.81 CYP24A1 (0.33)
SCHEMBL8876629 0.81 CYP24A1 (0.33)
SCHEMBL8876639 0.80 APP (0.32) KMT2AHSP90AA1POLB
SCHEMBL8874714 0.79 KMT2A (0.38) KMT2AHSP90AA1POLBCTDSP1KDM4E
SCHEMBL8874702 0.79 KMT2A (0.38) KMT2AHSP90AA1POLBCTDSP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5633373-A Enantioselective synthesis of antifolates ELI LILLY AND COMPANY (US) 1997-05-27 US disclosed
EP-0407212-B1 Enantioselective synthesis of antifolates LILLY CO ELI (US) 1996-05-22 EP disclosed
US-5516776-A Enantioselective synthesis of antifolates ELI LILLY AND COMPANY (US) 1996-05-14 US disclosed
US-5159090-A Enantioselective synthesis of antifolates ELI LILLY AND COMPANY (US) 1992-10-27 US disclosed
US-5008391-A Enantioselective synthesis of antifolates ELI LILLY AND COMPANY (US) 1991-04-16 US disclosed
EP-0407212-A1 Enantioselective synthesis of antifolates ELI LILLY AND COMPANY (US) 1991-01-09 EP disclosed