SCHEMBL8875258

SCHEMBL8875258

Cc1cc(CCCOc2c(Cl)cc(C(=N)NO)cc2Cl)on1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
HDAC6 Q9UBN7 4/20 0.42
HDAC4 P56524 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC11 Q96DB2 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC9 Q9UKV0 1/20 0.35
HDAC5 Q9UQL6 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
IGF1R P08069 4/20 0.33
FGFR1 P11362 4/20 0.33
KDR P35968 4/20 0.33
ALDH1A1 P00352 2/20 0.33
INSR P06213 1/20 0.33
VHL P40337 1/20 0.32
PLAU P00749 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8874123 0.94 NR1I2 (0.47) NR1I2CYP3A4CYP2D6HDAC6HDAC4
SCHEMBL8138666 0.88 NR1I2 (0.54) NR1I2CYP3A4CYP2D6HDAC6MEN1
SCHEMBL8875413 0.86 NR1I2 (0.47) NR1I2CYP3A4CYP2D6HDAC6MEN1
SCHEMBL8130660 0.85 CYP3A4 (0.43) NR1I2CYP3A4CYP2D6HDAC6MEN1
SCHEMBL9176420 0.83 NR1I2 (0.49) NR1I2CYP3A4CYP2D6HDAC6MEN1
SCHEMBL10413141 0.82 PLAU (0.51) NR1I2CYP3A4CYP2D6HDAC6MEN1
SCHEMBL8876078 0.81 NR1I2 (0.43) NR1I2CYP3A4CYP2D6HDAC6MEN1
SCHEMBL8876220 0.81 HDAC6 (0.46) NR1I2CYP3A4CYP2D6HDAC6MEN1
SCHEMBL10413619 0.79 NR1I2 (0.44) NR1I2CYP3A4CYP2D6HDAC6MEN1
SCHEMBL8875264 0.79 NR1I2 (0.44) NR1I2CYP3A4CYP2D6HDAC6MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5643929-A TREATMENT OF PICORNAVIRAL OR RHINOVIRUS AND CHEMICAL INTERMEDIATES SANOFI WINTHROP, INC. (US) 1997-07-01 US disclosed
US-5349068-A 1,2,4-oxadiazolyl-phenoxyalkylisoxazoles and their use as antiviral agents STERLING WINTHROP INC. (US) 1994-09-20 US disclosed