SCHEMBL8875413

SCHEMBL8875413

Cc1cc(CCCOc2c(F)cc(C(=N)NO)cc2F)on1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
IGF1R P08069 4/20 0.35
FGFR1 P11362 4/20 0.35
KDR P35968 4/20 0.35
INSR P06213 2/20 0.35
HDAC6 Q9UBN7 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
ALDH1A1 P00352 1/20 0.33
VHL P40337 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
GAA P10253 1/20 0.32
VRK1 Q99986 2/20 0.31
ROCK2 O75116 1/20 0.31
CSNK1D P48730 1/20 0.31
CSNK1E P49674 1/20 0.31
RPS6KA3 P51812 1/20 0.31
RPS6KA6 Q9UK32 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9176420 0.94 NR1I2 (0.49) NR1I2CYP3A4CYP2D6IGF1RFGFR1
SCHEMBL8876078 0.92 NR1I2 (0.43) NR1I2CYP3A4CYP2D6IGF1RFGFR1
SCHEMBL8138666 0.88 NR1I2 (0.54) NR1I2CYP3A4CYP2D6IGF1RFGFR1
SCHEMBL8875258 0.86 NR1I2 (0.44) NR1I2CYP3A4CYP2D6IGF1RFGFR1
SCHEMBL8130660 0.85 CYP3A4 (0.43) NR1I2CYP3A4CYP2D6IGF1RFGFR1
SCHEMBL8874123 0.83 NR1I2 (0.47) NR1I2CYP3A4CYP2D6IGF1RFGFR1
SCHEMBL8876220 0.81 HDAC6 (0.46) NR1I2CYP3A4CYP2D6IGF1RFGFR1
SCHEMBL8875424 0.79 NR1I2 (0.47) NR1I2CYP3A4CYP2D6IGF1RFGFR1
SCHEMBL8875008 0.78 NR1I2 (0.41) NR1I2CYP3A4CYP2D6IGF1RFGFR1
SCHEMBL9862923 0.78 NR1I2 (0.45) NR1I2CYP3A4CYP2D6MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5643929-A TREATMENT OF PICORNAVIRAL OR RHINOVIRUS AND CHEMICAL INTERMEDIATES SANOFI WINTHROP, INC. (US) 1997-07-01 US disclosed
US-5464848-A 1,2,4-oxadiazolyl-phenoxyalkylisoxazoles and their use as antiviral agents STERLING WINTHROP INC. (US) 1995-11-07 US disclosed
US-5349068-A 1,2,4-oxadiazolyl-phenoxyalkylisoxazoles and their use as antiviral agents STERLING WINTHROP INC. (US) 1994-09-20 US disclosed