SCHEMBL8875951

SCHEMBL8875951

C#CC(C(=O)Oc1c(-c2ccc(F)cc2)nc2ccccc2c1C(C)C)(C(C)O)[PH](=O)OC

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 4/20 0.53
TACR3 P29371 5/20 0.38
DHODH Q02127 3/20 0.37
PDE10A Q9Y233 1/20 0.33
SCN9A Q15858 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8877114 0.91 HMGCR (0.52) HMGCRTACR3DHODHPDE10ASCN9A
SCHEMBL8900673 0.86 HMGCR (0.48) HMGCRTACR3DHODHPDE10ASCN9A
SCHEMBL8877778 0.85 HMGCR (0.38) HMGCR
SCHEMBL8901358 0.83 HMGCR (0.37) HMGCR
SCHEMBL8877730 0.83 HMGCR (0.38) HMGCRDHODH
SCHEMBL8876883 0.82 HMGCR (0.44) HMGCRTACR3DHODHPDE10ASCN9A
SCHEMBL8899623 0.81 HMGCR (0.34) HMGCR
SCHEMBL8899571 0.81 HMGCR (0.34) HMGCR
SCHEMBL8877820 0.81 HMGCR (0.41) HMGCRDHODHPDE10A
SCHEMBL8876699 0.79 GCGR (0.37) HMGCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691322-A Quinoline and pyridine anchors for HMG-CoA reductase inhibitors E.R. SQUIBB & SONS, INC. (US) 1997-11-25 US disclosed
US-5686433-A CHOLESTEROL BIOSYNTHESIS INHIBITION E.R. SQUIBB & SONS, INC. (US) 1997-11-11 US disclosed