SCHEMBL8876345

SCHEMBL8876345

CC(C)c1nc(C(c2ccccc2)c2ccccc2)cc(-c2ccc(F)cc2)c1C=C(Br)Br

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GCGR P47871 3/20 0.41
HMGCR P04035 5/20 0.40
PTGS2 P35354 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8876861 0.87 GCGR (0.46) GCGRHMGCR
SCHEMBL8878730 0.85 HMGCR (0.42) GCGRHMGCRPTGS2
SCHEMBL8876495 0.84 HMGCR (0.54) GCGRHMGCR
SCHEMBL8952722 0.83 HMGCR (0.41) GCGRHMGCR
SCHEMBL8877967 0.80 HMGCR (0.52) GCGRHMGCR
SCHEMBL8877450 0.79 GCGR (0.50) GCGRHMGCR
SCHEMBL8878764 0.79 HMGCR (0.44) GCGRHMGCR
SCHEMBL8952718 0.78 HMGCR (0.43) GCGRHMGCRPTGDR2
SCHEMBL8877751 0.78 DHODH (0.42) GCGRPTGDR2
SCHEMBL8876862 0.78 HMGCR (0.42) GCGRHMGCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691322-A Quinoline and pyridine anchors for HMG-CoA reductase inhibitors E.R. SQUIBB & SONS, INC. (US) 1997-11-25 US disclosed
US-5686433-A CHOLESTEROL BIOSYNTHESIS INHIBITION E.R. SQUIBB & SONS, INC. (US) 1997-11-11 US disclosed