SCHEMBL8876455

SCHEMBL8876455

COc1ccccc1N1CCN(CCCNc2cccc3c(=O)c(C)c(-c4ccccc4)oc23)CC1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 8/20 0.75
ADRA1D P25100 7/20 0.75
ADRA1B P35368 7/20 0.75
HTR1A P08908 7/20 0.75
ALDH1A1 P00352 1/20 0.61
LMNA P02545 1/20 0.61
ADRA2A P08913 2/20 0.54
CYP3A4 P08684 1/20 0.54
ADRA2B P18089 1/20 0.54
ADRA2C P18825 1/20 0.54
PMP22 Q01453 1/20 0.54
HIF1A Q16665 1/20 0.54
DRD3 P35462 3/20 0.51
DRD2 P14416 2/20 0.51
DRD1 P21728 1/20 0.51
DRD4 P21917 1/20 0.51
DRD5 P21918 1/20 0.51
HTR2A P28223 1/20 0.51
FAAH O00519 2/20 0.51
CNR1 P21554 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL27348716 0.99 ADRA1A (0.74) ADRA1AADRA1DADRA1BHTR1AALDH1A1
SCHEMBL8875934 0.97 HTR1A (0.71) ADRA1AADRA1DADRA1BHTR1AALDH1A1
Hydrochloric Acid SCHEMBL8875713 0.96 HTR1A (0.69) ADRA1AADRA1DADRA1BHTR1AALDH1A1
Hydrochloric Acid SCHEMBL8875715 0.96 HTR1A (0.69) ADRA1AADRA1DADRA1BHTR1AALDH1A1
SCHEMBL8877818 0.95 HTR1A (0.69) ADRA1AADRA1DADRA1BHTR1AALDH1A1
Hydrochloric Acid SCHEMBL8875648 0.94 HTR1A (0.69) ADRA1AADRA1DADRA1BHTR1AALDH1A1
SCHEMBL8875435 0.87 HTR1A (0.71) ADRA1AADRA1DADRA1BHTR1AALDH1A1
SCHEMBL8876154 0.87 ADRA1A (0.73) ADRA1AADRA1DADRA1BHTR1AALDH1A1
SCHEMBL8876505 0.86 HTR1A (0.71) ADRA1AADRA1DADRA1BHTR1AALDH1A1
Hydrochloric Acid SCHEMBL8876536 0.86 ADRA1A (0.72) ADRA1AADRA1DADRA1BHTR1AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1040434-C Heterobicyclic compounds RECORDATI CHEM PHARM (CH) 1998-10-28 CN claimed
US-5605896-A Bicyclic heterocyclic derivatives having α1 adrenergic and 5HT1A activities RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1997-02-25 US claimed
US-5403842-A Adrenergic blocking and antiserotonine agents; urogenital disorders including spasms of the urethral tract and prostrate problems RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1995-04-04 US claimed
EP-0558245-A1 Heterobicyclic compounds as antagogists of alpha-1 adrenergic and SHT1A receptors RECORDATI S.A. CHEMICAL and PHARMACEUTICAL COMPANY (CH) 1993-09-01 EP claimed