SCHEMBL8876804

SCHEMBL8876804

CCOC(=O)c1cccc2c(=O)c(C)c(-c3ccc(Oc4ccccc4)cc3)oc12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.60
LMNA P02545 6/20 0.60
KDM4E B2RXH2 2/20 0.60
CYP1A2 P05177 1/20 0.60
CHRM2 P08172 1/20 0.60
CYP3A4 P08684 1/20 0.60
HTR1A P08908 1/20 0.60
ADRA2A P08913 1/20 0.60
ADORA3 P0DMS8 1/20 0.60
CYP2D6 P10635 1/20 0.60
CHRM1 P11229 1/20 0.60
ACHE P22303 1/20 0.60
SLC6A2 P23975 1/20 0.60
PDE4A P27815 1/20 0.60
ADRA1A P35348 1/20 0.60
OPRM1 P35372 1/20 0.60
DRD3 P35462 1/20 0.60
KCNH2 Q12809 1/20 0.60
HRH3 Q9Y5N1 1/20 0.60
MAPT P10636 5/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8875460 0.91 ALDH1A1 (0.67) ALDH1A1LMNAKDM4ECYP1A2CHRM2
SCHEMBL8878647 0.91 ALDH1A1 (0.69) ALDH1A1LMNAKDM4ECYP1A2CHRM2
SCHEMBL8877000 0.89 ALDH1A1 (0.56) ALDH1A1LMNAKDM4ECYP1A2CHRM2
SCHEMBL27345512 0.89 MAPT (0.59) ALDH1A1LMNAKDM4ECYP1A2CHRM2
SCHEMBL8875613 0.88 CYSLTR1 (0.61) ALDH1A1LMNAKDM4ECYP1A2CHRM2
SCHEMBL27352550 0.88 LMNA (0.68) ALDH1A1LMNAKDM4ECYP1A2CHRM2
SCHEMBL8876105 0.87 MAPT (0.62) ALDH1A1LMNAKDM4ECYP1A2CHRM2
SCHEMBL10842166 0.87 LMNA (0.58) ALDH1A1LMNAKDM4ECYP1A2CHRM2
SCHEMBL10841682 0.86 LMNA (0.57) ALDH1A1LMNAKDM4ECYP1A2CHRM2
SCHEMBL8875388 0.86 MAPT (0.69) ALDH1A1LMNAKDM4ECYP1A2CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1040434-C Heterobicyclic compounds RECORDATI CHEM PHARM (CH) 1998-10-28 CN disclosed
US-5605896-A Bicyclic heterocyclic derivatives having α1 adrenergic and 5HT1A activities RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1997-02-25 US disclosed
US-5474994-A Treating hypertension, urethral and lower urinary tract contractions RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1995-12-12 US disclosed
CN-1079738-A Heterobicyclic compounds RECORDATI CHEM PHARM (CH) 1993-12-22 CN disclosed
WO-1993017007-A1 HETEROBICYCLIC COMPOUNDS RECORDATI INDUSTRIA CHIMICA E FARMACEUTICA S.P.A. (IT) 1993-09-02 WO disclosed
EP-0558245-A1 Heterobicyclic compounds as antagogists of alpha-1 adrenergic and SHT1A receptors RECORDATI S.A. CHEMICAL and PHARMACEUTICAL COMPANY (CH) 1993-09-01 EP disclosed