SCHEMBL8877083

SCHEMBL8877083

CCOC(=O)C1CCC(C)N1C(=O)Cc1ccc(Cl)cc1Cl

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.45
MAPK1 P28482 1/20 0.45
RECQL P46063 1/20 0.45
P2RX7 Q99572 7/20 0.43
KMT2A Q03164 3/20 0.42
ERCC1 P07992 1/20 0.42
ERCC4 Q92889 1/20 0.42
SIGMAR1 Q99720 1/20 0.41
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8876049 0.94 TSHR (0.48) TSHRMAPK1RECQLP2RX7KMT2A
SCHEMBL8875758 0.87 TSHR (0.41) TSHRMAPK1RECQLP2RX7KMT2A
SCHEMBL8877223 0.84 TSHR (0.46) TSHRMAPK1RECQLP2RX7KMT2A
SCHEMBL8876722 0.83 TSHR (0.44) TSHRMAPK1RECQLP2RX7KMT2A
SCHEMBL8313154 0.83 KMT2A (0.41) TSHRP2RX7KMT2AERCC1ERCC4
SCHEMBL8876826 0.83 TSHR (0.46) TSHRMAPK1RECQLP2RX7KMT2A
SCHEMBL8877202 0.82 P2RX7 (0.43) TSHRMAPK1RECQLP2RX7KMT2A
SCHEMBL8875634 0.81 KMT2A (0.42) TSHRMAPK1RECQLKMT2AERCC1
SCHEMBL8876904 0.81 KMT2A (0.54) TSHRP2RX7KMT2AMEN1ALDH1A1
SCHEMBL8875647 0.80 TSHR (0.45) TSHRMAPK1RECQLP2RX7KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4338390-A None JP disclosed
US-5693663-A PESTICIDES; HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 1997-12-02 US disclosed
US-5585384-A 1-OXY-FUNCTIONAL GROUP-2-ALKYLARYL-3-OXO-PYRROLIZINES; INSECTICIDES; NEMATOCIDES; HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 1996-12-17 US disclosed
US-5288874-A Insecticides, miticides BAYER AKTIENGESELLSCHAFT (DE) 1994-02-22 US disclosed
JP-H04338390-A BICYCLIC 3-ARYL-PYRROLIDIN-2,4-DIONE DERIVATIVE BAYER AG 1992-11-25 JP disclosed