SCHEMBL8877685

SCHEMBL8877685

O=C(O)C12CC(c3ccc(Cl)cc31)c1ccc(Cl)cc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 2/20 0.38
HSD11B1 P28845 1/20 0.36
KDM1A O60341 2/20 0.35
DRD1 P21728 1/20 0.34
ALDH1A1 P00352 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
TP53 P04637 1/20 0.34
TSHR P16473 1/20 0.34
CASP1 P29466 1/20 0.34
NOTUM Q6P988 1/20 0.34
HSP90AA1 P07900 1/20 0.34
PRKAB2 O43741 1/20 0.34
PRKAG1 P54619 1/20 0.34
PRKAA2 P54646 1/20 0.34
PRKAA1 Q13131 1/20 0.34
PRKAG3 Q9UGI9 1/20 0.34
PRKAG2 Q9UGJ0 1/20 0.34
PRKAB1 Q9Y478 1/20 0.34
KCNK2 O95069 1/20 0.33
CA1 P00915 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9035580 0.93 DRD1 (0.38) AKR1B1HSD11B1DRD1ALDH1A1MEN1
SCHEMBL8601902 0.93 DRD1 (0.38) AKR1B1HSD11B1DRD1ALDH1A1MEN1
SCHEMBL8601315 0.93 DRD1 (0.38) AKR1B1HSD11B1DRD1ALDH1A1MEN1
SCHEMBL8878875 0.93 AKR1B1 (0.34) AKR1B1HSD11B1DRD1TSHRCA1
SCHEMBL8602565 0.93 DRD1 (0.38) AKR1B1HSD11B1DRD1ALDH1A1MEN1
SCHEMBL9035567 0.93 DRD1 (0.38) AKR1B1HSD11B1DRD1ALDH1A1MEN1
SCHEMBL8601899 0.93 DRD1 (0.38) AKR1B1HSD11B1DRD1ALDH1A1MEN1
SCHEMBL8602566 0.93 DRD1 (0.38) AKR1B1HSD11B1DRD1ALDH1A1MEN1
SCHEMBL8876907 0.91 AKR1B1 (0.34) AKR1B1HSD11B1KDM1ADRD1ALDH1A1
SCHEMBL8875582 0.88 CDYL (0.40) ALDH1A1SMN1; SMN2TSHRMEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5681840-A ANTIDOPAMINERGIC AGENTS ZENECA LIMITED (GB) 1997-10-28 US disclosed
EP-0533344-B1 Methanoanthracenes as dopamine antagonists ZENECA LTD (GB) 1996-10-16 EP disclosed
US-5512575-A ANTISEROTONINE AGENT ZENECA LIMITED (GB) 1996-04-30 US disclosed
EP-0533344-A1 Methanoanthracenes as dopamine antagonists ZENECA LIMITED (GB) 1993-03-24 EP disclosed