SCHEMBL8877845

SCHEMBL8877845

CC(C)C(=O)C(C(=O)O)C(CC(=O)C(c1ccccc1)c1ccccc1)c1ccc(F)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.41
NPC1 O15118 1/20 0.41
PDPK1 O15530 2/20 0.40
ALDH1A1 P00352 3/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2D6 P10635 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
KDM4E B2RXH2 1/20 0.39
KLK7 P49862 3/20 0.38
POLB P06746 1/20 0.38
LMNA P02545 2/20 0.37
HTT P42858 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
USP2 O75604 1/20 0.37
HPGD P15428 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MEN1 O00255 1/20 0.37
CYP1A2 P05177 1/20 0.37
CRHBP P24387 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8877170 0.88 MME (0.40) NPC1PDPK1ALDH1A1KDM4ELMNA
SCHEMBL8878618 0.84 PDPK1 (0.51) TDP1NPC1PDPK1ALDH1A1KDM4E
SCHEMBL8878251 0.82 LMNA (0.37) NPC1PDPK1ALDH1A1KDM4ELMNA
SCHEMBL8876896 0.79 PDPK1 (0.41) TDP1NPC1PDPK1ALDH1A1KDM4E
SCHEMBL8876550 0.79 PDPK1 (0.36) NPC1PDPK1ALDH1A1KDM4ELMNA
SCHEMBL8878459 0.76 PDPK1 (0.40) TDP1PDPK1ALDH1A1CYP3A4CYP2D6
SCHEMBL9857098 0.76 PDPK1 (0.55) PDPK1ALDH1A1CYP3A4CYP2D6KDM4E
SCHEMBL917627 0.73 NPC1 (0.48) TDP1NPC1ALDH1A1CYP3A4CYP2D6
SCHEMBL9655539 0.73 NPC1 (0.41) TDP1NPC1ALDH1A1CYP2D6KDM4E
SCHEMBL2142907 0.72 PDPK1 (0.63) TDP1PDPK1ALDH1A1LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691322-A Quinoline and pyridine anchors for HMG-CoA reductase inhibitors E.R. SQUIBB & SONS, INC. (US) 1997-11-25 US disclosed
US-5686433-A CHOLESTEROL BIOSYNTHESIS INHIBITION E.R. SQUIBB & SONS, INC. (US) 1997-11-11 US disclosed
US-5506219-A ANTICHOLESTEROL AND ANTILIPEMIC AGENTS E. R. SQUIBB & SONS, INC. (US) 1996-04-09 US disclosed