SCHEMBL8878029

SCHEMBL8878029

Cc1c(CCC(=O)O)c2cc(Br)ccc2n1Cc1ccc(Br)cc1

nearest known ligand 0.80

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.62
PLA2G2A P14555 6/20 0.59
THRA P10827 1/20 0.53
THRB P10828 1/20 0.53
PTGES O14684 1/20 0.51
ALOX5 P09917 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8877434 0.94 PLA2G2A (0.62) PTGS2PLA2G2ATHRATHRB
SCHEMBL3242276 0.93 PTGS2 (0.60) PTGS2PLA2G2ATHRATHRBPTGES
SCHEMBL3246296 0.92 PTGS2 (0.59) PTGS2PLA2G2ATHRATHRBPTGES
SCHEMBL3246589 0.89 PTGS2 (0.80) PTGS2PLA2G2A
SCHEMBL8876716 0.89 PLA2G2A (0.59) PTGS2PLA2G2ATHRATHRBPTGES
SCHEMBL9230125 0.88 PTGS2 (0.79) PTGS2PLA2G2APTGESALOX5
SCHEMBL8876622 0.87 PLA2G2A (0.60) PTGS2PLA2G2ATHRATHRBPTGES
SCHEMBL8878924 0.86 PLA2G2A (0.59) PTGS2PLA2G2ATHRATHRBPTGES
SCHEMBL7196880 0.83 PTGS2 (0.79) PTGS2PLA2G2A
SCHEMBL8878256 0.81 PLA2G2A (0.58) PTGS2PLA2G2APTGESALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996037469-A1 N-BENZYLINDOL-3-YL PROPANIC ACID DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS MERCK FROSST CANADA INC. (CA) 1996-11-28 WO claimed
US-5604253-A ANTIINFLAMMATORY AGENTS, ANALGESICS, ANTIPYRETICS MERCK FROSST CANADA, INC. (CA) 1997-02-18 US disclosed
WO-1996037469-A1 N-BENZYLINDOL-3-YL PROPANIC ACID DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS MERCK FROSST CANADA INC. (CA) 1996-11-28 WO disclosed