SCHEMBL8878474

SCHEMBL8878474

CC(C)c1nc(C(C)(C)C)cc(-c2ccc(F)cc2)c1C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 1/20 0.48
SQOR Q9Y6N5 1/20 0.43
GCGR P47871 4/20 0.43
DHODH Q02127 3/20 0.40
DPP4 P27487 1/20 0.39
DPP8 Q6V1X1 1/20 0.39
DPP9 Q86TI2 1/20 0.39
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
KMT2A Q03164 1/20 0.38
FABP3 P05413 1/20 0.37
FABP4 P15090 1/20 0.37
FABP5 Q01469 1/20 0.37
PPARA Q07869 1/20 0.37
DHFR P00374 1/20 0.37
ALKBH5 Q6P6C2 1/20 0.37
AKR1C3 P42330 1/20 0.36
AKR1C2 P52895 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8876825 0.83 PPARA (0.46) HMGCRGCGRDHODHMEN1NPC1
SCHEMBL8880943 0.83 GCGR (0.45) GCGRDHODHFABP3FABP4FABP5
SCHEMBL8879993 0.81 HMGCR (0.49) HMGCRSQORGCGRDHODHFABP3
SCHEMBL8878856 0.80 GCGR (0.46) HMGCRGCGRFABP3FABP4FABP5
SCHEMBL8879135 0.79 GCGR (0.54) HMGCRGCGR
SCHEMBL8878217 0.78 HMGCR (0.57) HMGCRSQORGCGR
SCHEMBL8878154 0.77 DHODH (0.44) HMGCRSQORGCGRDHODHFABP3
SCHEMBL8877751 0.77 DHODH (0.42) GCGRDHODHFABP3FABP4FABP5
SCHEMBL8875727 0.76 HMGCR (0.57) HMGCRSQORGCGR
SCHEMBL8875731 0.76 HMGCR (0.57) HMGCRSQORGCGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691322-A Quinoline and pyridine anchors for HMG-CoA reductase inhibitors E.R. SQUIBB & SONS, INC. (US) 1997-11-25 US disclosed
US-5686433-A CHOLESTEROL BIOSYNTHESIS INHIBITION E.R. SQUIBB & SONS, INC. (US) 1997-11-11 US disclosed
US-5506219-A ANTICHOLESTEROL AND ANTILIPEMIC AGENTS E. R. SQUIBB & SONS, INC. (US) 1996-04-09 US disclosed