SCHEMBL8878154

SCHEMBL8878154

Cc1ccccc1-c1cc(-c2ccc(F)cc2)c(C(=O)O)c(C(C)C)n1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 4/20 0.44
DHFR P00374 1/20 0.44
ALKBH5 Q6P6C2 1/20 0.44
HMGCR P04035 3/20 0.42
GCGR P47871 1/20 0.41
LDHA P00338 1/20 0.40
PDE10A Q9Y233 1/20 0.40
FABP3 P05413 1/20 0.40
FABP4 P15090 1/20 0.40
FABP5 Q01469 1/20 0.40
SQOR Q9Y6N5 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8879993 0.88 HMGCR (0.49) DHODHHMGCRGCGRFABP3FABP4
SCHEMBL8876808 0.86 MEN1 (0.46) DHODHDHFRALKBH5HMGCRFABP3
SCHEMBL8877871 0.85 PTGDR2 (0.42) DHODHDHFRALKBH5HMGCRGCGR
SCHEMBL8876825 0.85 PPARA (0.46) DHODHDHFRALKBH5HMGCRGCGR
SCHEMBL8878856 0.81 GCGR (0.46) HMGCRGCGRFABP3FABP4FABP5
SCHEMBL8877443 0.81 GCGR (0.54) HMGCRGCGR
SCHEMBL8880943 0.80 GCGR (0.45) DHODHDHFRALKBH5GCGRFABP3
SCHEMBL8876796 0.80 HMGCR (0.46) HMGCRGCGR
SCHEMBL8877509 0.79 MEN1 (0.49) DHODHGCGR
SCHEMBL8877954 0.79 DHODH (0.43) DHODHDHFRALKBH5HMGCRLDHA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691322-A Quinoline and pyridine anchors for HMG-CoA reductase inhibitors E.R. SQUIBB & SONS, INC. (US) 1997-11-25 US disclosed
US-5686433-A CHOLESTEROL BIOSYNTHESIS INHIBITION E.R. SQUIBB & SONS, INC. (US) 1997-11-11 US disclosed
US-5506219-A ANTICHOLESTEROL AND ANTILIPEMIC AGENTS E. R. SQUIBB & SONS, INC. (US) 1996-04-09 US disclosed