SCHEMBL8878621

SCHEMBL8878621

C/C=C(\C)C(=O)c1cc(-c2ccccc2)no1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.60
SMN1; SMN2 Q16637 3/20 0.60
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
ALDH1A1 P00352 1/20 0.49
NOTUM Q6P988 2/20 0.47
NPC1 O15118 4/20 0.46
MAPT P10636 2/20 0.46
CYP2C19 P33261 2/20 0.46
CYP1A2 P05177 1/20 0.46
KDM4E B2RXH2 1/20 0.46
PTPN1 P18031 2/20 0.44
RXFP1 Q9HBX9 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
TSHR P16473 1/20 0.42
CASP3 P42574 1/20 0.42
SENP8 Q96LD8 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8878628 1.00 RAB9A (0.60) RAB9ASMN1; SMN2MEN1KMT2AALDH1A1
SCHEMBL4805 0.82 RAB9A (0.69) RAB9ASMN1; SMN2MEN1KMT2AALDH1A1
SCHEMBL9371664 0.80 RAB9A (0.60) RAB9ASMN1; SMN2MEN1KMT2AALDH1A1
SCHEMBL8878334 0.80 SMN1; SMN2 (0.65) RAB9ASMN1; SMN2MEN1KMT2AALDH1A1
SCHEMBL8975518 0.79 SMN1; SMN2 (0.57) RAB9ASMN1; SMN2MEN1KMT2AALDH1A1
SCHEMBL8879679 0.79 RAB9A (0.60) RAB9ASMN1; SMN2MEN1KMT2AALDH1A1
SCHEMBL8879700 0.79 RAB9A (0.60) RAB9ASMN1; SMN2MEN1KMT2AALDH1A1
SCHEMBL28091339 0.79 RAB9A (0.68) RAB9ASMN1; SMN2MEN1KMT2AALDH1A1
SCHEMBL212382 0.79 RAB9A (0.68) RAB9ASMN1; SMN2MEN1KMT2AALDH1A1
SCHEMBL1435521 0.78 RAB9A (0.59) RAB9ASMN1; SMN2MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5602160-A MUSCLE RELAXANT MITSUI TOATSU CHEMICALS INCORPORATED (JP) 1997-02-11 US disclosed
US-5498619-A MUSCLE RELAXANTS, POLLAKIUREA CURING AGENTS AND MUSCLE SPASMS MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1996-03-12 US disclosed
EP-0414391-B1 Aminoketone derivatives and use thereof MITSUI TOATSU CHEMICALS (JP) 1995-03-15 EP disclosed
US-5338857-A Muscle relaxant MITSUI TOATSU CHEMICALS INCORPORATED (JP) 1994-08-16 US disclosed
EP-0414391-A2 Aminoketone derivatives and use thereof MITSUI TOATSU CHEMICALS, Inc. (JP) 1991-02-27 EP disclosed