SCHEMBL8879520

SCHEMBL8879520

Cc1cc(C)nc(NCC(O)CO)n1

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.60
SMN1; SMN2 Q16637 1/20 0.57
NPSR1 Q6W5P4 1/20 0.55
KMT2A Q03164 2/20 0.55
MEN1 O00255 1/20 0.55
GAA P10253 1/20 0.55
MAPK1 P28482 1/20 0.55
KDM4E B2RXH2 1/20 0.46
IDH2 P48735 3/20 0.46
CYP1A2 P05177 1/20 0.45
ALPL P05186 1/20 0.44
ALPG P10696 1/20 0.44
PLAA Q9Y263 1/20 0.44
MAPT P10636 2/20 0.40
ESR1 P03372 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1692066 0.82 IDH2 (0.50) LMNASMN1; SMN2NPSR1IDH2ESR1
SCHEMBL16015949 0.81 IDH2 (0.44) LMNASMN1; SMN2NPSR1GAAIDH2
SCHEMBL9114392 0.77 CYP1A2 (0.54) LMNASMN1; SMN2NPSR1GAACYP1A2
SCHEMBL12870821 0.76 ESR1 (0.64) LMNASMN1; SMN2NPSR1KMT2AMEN1
SCHEMBL12523522 0.74 P2RX3 (0.41) LMNASMN1; SMN2NPSR1IDH2CYP1A2
SCHEMBL16015948 0.74 IDH2 (0.37) LMNASMN1; SMN2NPSR1IDH2CYP1A2
SCHEMBL1691640 0.73 IDH2 (0.44) LMNASMN1; SMN2IDH2
SCHEMBL1692063 0.73 IDH2 (0.41) LMNASMN1; SMN2IDH2
SCHEMBL13034405 0.72 KMT2A (0.96) KMT2AMEN1GAAMAPK1KDM4E
SCHEMBL11403184 0.71 LMNA (0.47) LMNASMN1; SMN2NPSR1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5616708-A CHEMICAL INTERMEDIATES SHELL RESEARCH LIMITED (GB) 1997-04-01 US disclosed
US-5599818-A A 3-(PYRIMIDIN-2-YL-AMINOALKYL-)-1-OXA OR 1,4-DIOXASPIRO-4.(5 TO 8)ALKANE(9 TO 12 C'S); PATHOGENIC FUNGI; CROPS SHELL RESEARCH LIMITED (GB) 1997-02-04 US disclosed
US-5462944-A Applying spiroheterocyclic compounds SHELL RESEARCH LIMITED (GB) 1995-10-31 US disclosed
EP-0623613-A1 Fungicidal spiroheterocyclic compounds SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1994-11-09 EP disclosed