SCHEMBL8880302

SCHEMBL8880302

CC(C)(C)ON(C=O)C(CO)c1ccc(Cl)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
AOC3 Q16853 2/20 0.33
MAPT P10636 2/20 0.32
ALDH1A1 P00352 1/20 0.32
SLC6A4 P31645 1/20 0.32
KCNH2 Q12809 1/20 0.32
FFAR2 O15552 1/20 0.32
BRD4 O60885 1/20 0.32
GRIN2D O15399 1/20 0.31
GRIN3B O60391 1/20 0.31
GRIN1 Q05586 1/20 0.31
GRIN2A Q12879 1/20 0.31
GRIN2B Q13224 1/20 0.31
GRIN2C Q14957 1/20 0.31
GRIN3A Q8TCU5 1/20 0.31
CYP1A2 P05177 1/20 0.31
THRB P10828 1/20 0.31
PMP22 Q01453 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6184942 0.85 NR1H2 (0.36) LMNAMAPTALDH1A1
SCHEMBL4728453 0.78 SLC6A2 (0.35) LMNAMAPTALDH1A1SLC6A4KCNH2
SCHEMBL18222240 0.69 SLC6A4 (0.38) LMNAMAPTSLC6A4BRD4CYP1A2
SCHEMBL7343190 0.69 KCNA5 (0.45) SMN1; SMN2MAPTALDH1A1
SCHEMBL1649228 0.68
SCHEMBL629756 0.68
SCHEMBL3977769 0.67 MT-CO2 (0.38) SMN1; SMN2MAPTALDH1A1
SCHEMBL21979520 0.66 AOC3 (0.41) LMNAAOC3ALDH1A1BRD4CYP1A2
SCHEMBL20660981 0.66 AOC3 (0.41) LMNAAOC3ALDH1A1BRD4CYP1A2
SCHEMBL21979530 0.66 AOC3 (0.41) LMNAAOC3ALDH1A1BRD4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5610183-A Phenylglycine derivatives pharmaceutical compositions containing them and their use in therapy MERCK, SHARP & DOHME LTD. (GB) 1997-03-11 US disclosed
EP-0593615-A1 AROMATIC COMPOUNDS, COMPOSITIONS CONTAINING THEM AND THEIR USE IN THERAPY. MERCK SHARP & DOHME (GB) 1994-04-27 EP disclosed
WO-1993001165-A2 AROMATIC COMPOUNDS, COMPOSITIONS CONTAINING THEM AND THEIR USE IN THERAPY MERCK SHARP & DOHME LIMITED (GB) 1993-01-21 WO disclosed