SCHEMBL8880862

SCHEMBL8880862

C#CCN1CCN(c2cccc3c2CCC(=O)N3)CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 14/20 0.53
DRD4 P21917 2/20 0.52
DRD3 P35462 2/20 0.52
SCN1A P35498 1/20 0.48
SCN5A Q14524 1/20 0.48
SCN9A Q15858 1/20 0.48
HTR1A P08908 5/20 0.47
SLC6A4 P31645 4/20 0.47
HTR1D P28221 3/20 0.47
HTR1B P28222 3/20 0.47
KCNH2 Q12809 3/20 0.47
HTR2A P28223 3/20 0.41
HTR3E A5X5Y0 1/20 0.40
MEN1 O00255 1/20 0.40
MLNR O43193 1/20 0.40
HTR3B O95264 1/20 0.40
ABCB11 O95342 1/20 0.40
ESR1 P03372 1/20 0.40
PGR P06401 1/20 0.40
ADRB2 P07550 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11198122 0.82 DRD2 (0.55) DRD2DRD4DRD3SCN1ASCN5A
Hydrochloric Acid SCHEMBL11203073 0.79 DRD2 (0.78) DRD2DRD4DRD3SCN1ASCN5A
SCHEMBL11194827 0.77 DRD2 (0.49) DRD2DRD4DRD3SCN1ASCN5A
SCHEMBL11199800 0.77 DRD2 (0.60) DRD2DRD4DRD3SCN1ASCN5A
SCHEMBL11197104 0.76 DRD2 (0.52) DRD2DRD4DRD3SCN1ASCN5A
Bromide SCHEMBL11196359 0.76 DRD2 (0.48) DRD2DRD4DRD3SCN1ASCN5A
Hydrochloric Acid SCHEMBL11204105 0.75 DRD2 (0.61) DRD2DRD4DRD3SCN1ASCN5A
Hydrochloric Acid SCHEMBL11196563 0.75 DRD2 (0.47) DRD2DRD4DRD3SCN1ASCN5A
SCHEMBL11201027 0.75 ALDH1A1 (0.52) DRD2DRD4DRD3SCN1ASCN5A
SCHEMBL11194927 0.75 DRD2 (0.60) DRD2DRD4DRD3SCN1ASCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691341-A ANTILEUKEMIA AGENT OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-11-25 US disclosed
EP-0623598-A1 APOPTOSIS REGULATOR OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-11-09 EP disclosed
US-4415572-A CARDIOTONIC AND INOTROPIC AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1983-11-15 US disclosed