SCHEMBL8881815

SCHEMBL8881815

CS(=O)(=O)OCC1(CN(Cc2ccccc2)Cc2ccccc2)CCN(Cc2ccccc2)C1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 11/20 0.48
CYP3A4 P08684 6/20 0.48
TSHR P16473 4/20 0.48
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
USP2 O75604 2/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
CXCR4 P61073 2/20 0.40
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
OPRM1 P35372 1/20 0.38
SIGMAR1 Q99720 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16197363 0.81 CYP2D6 (0.52) CYP2D6CYP3A4TSHRMEN1KMT2A
SCHEMBL8880097 0.79 CYP3A4 (0.43) CYP2D6CYP3A4TSHRMEN1KMT2A
SCHEMBL8881966 0.79 POLB (0.49) CYP3A4MEN1KMT2AALDH1A1OPRM1
SCHEMBL1290767 0.77 CYP2D6 (0.49) CYP2D6CYP3A4TSHRMEN1KMT2A
SCHEMBL9233359 0.74 POLB (0.54) CYP2D6CYP3A4TSHRMEN1KMT2A
SCHEMBL9228415 0.72 ALDH1A1 (0.58) CYP2D6MEN1KMT2AALDH1A1
SCHEMBL9232502 0.72 CYP2D6 (0.47) CYP2D6CYP3A4TSHRALDH1A1SIGMAR1
SCHEMBL9566488 0.71 CYP2D6 (0.48) CYP2D6CYP3A4TSHRMEN1KMT2A
SCHEMBL8883321 0.70 POLB (0.49) CYP2D6CYP3A4TSHRMEN1KMT2A
SCHEMBL8881229 0.70 HRH3 (0.47) CYP2D6CYP3A4TSHRMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5677316-A BACTERICIDES YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-10-14 US disclosed
EP-0677522-A1 8-METHOXYQUINOLONECARBOXYLIC ACID DERIVATIVE YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1995-10-18 EP disclosed