SCHEMBL8883641

SCHEMBL8883641

CC(C)CCOc1ccnc(C(=O)NC(=O)[C@H](C)N)c1O

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.40
EPHX2 P34913 1/20 0.36
MAPK1 P28482 1/20 0.35
XDH P47989 1/20 0.34
GALR3 O60755 1/20 0.33
HSP90AA1 P07900 1/20 0.33
TLR8 Q9NR97 1/20 0.33
MCHR1 Q99705 1/20 0.33
KDM4E B2RXH2 1/20 0.33
PPIA P62937 1/20 0.33
CARM1 Q86X55 1/20 0.33
PRMT6 Q96LA8 1/20 0.33
CYP19A1 P11511 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8883147 0.91 HTT (0.39) HTTEPHX2MAPK1XDHGALR3
SCHEMBL8883790 0.90 AAK1 (0.39) HTT
SCHEMBL8883362 0.89 IKBKB (0.38) HTTMAPK1KDM4ECARM1PRMT6
SCHEMBL8882922 0.89 IKBKB (0.38) HTTMAPK1KDM4ECARM1PRMT6
SCHEMBL8882551 0.88 LNPEP (0.36) HTTKDM4ECARM1PRMT6
SCHEMBL8884848 0.88 XIAP (0.42)
SCHEMBL8882517 0.88 LNPEP (0.36) HTTKDM4ECARM1PRMT6
SCHEMBL8881873 0.88 XIAP (0.42)
SCHEMBL8883971 0.88 CYP3A4 (0.35) HTTXDH
SCHEMBL8882669 0.87 PTPN1 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5620995-A Substituted heterocyclic carboxyamides, their preparation and their use as pharmaceuticals HOECHST AKTIENGESELLSCHAFT (DE) 1997-04-15 US disclosed