SCHEMBL8883147

SCHEMBL8883147

CC(C)CCOc1ccnc(C(=O)NC(=O)[C@@H](N)C(C)C)c1O

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.39
EPHX2 P34913 1/20 0.34
MAPK1 P28482 1/20 0.33
XDH P47989 1/20 0.33
KDM4E B2RXH2 1/20 0.32
GALR3 O60755 1/20 0.32
HSP90AA1 P07900 1/20 0.32
PPIA P62937 1/20 0.32
TLR8 Q9NR97 1/20 0.32
MCHR1 Q99705 1/20 0.32
CIT O14578 1/20 0.32
CYP19A1 P11511 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8883641 0.91 HTT (0.40) HTTEPHX2MAPK1XDHKDM4E
SCHEMBL8883790 0.88 AAK1 (0.39) HTTCIT
SCHEMBL8881773 0.84 HTT (0.40) HTTEPHX2MAPK1XDHKDM4E
SCHEMBL8883021 0.83 CIT (0.31) CIT
SCHEMBL8882386 0.82 LNPEP (0.36) MCHR1
SCHEMBL8779208 0.82 HTT (0.38) HTTEPHX2MAPK1XDHKDM4E
SCHEMBL8882922 0.80 IKBKB (0.38) HTTMAPK1KDM4ECIT
SCHEMBL8883362 0.80 IKBKB (0.38) HTTMAPK1KDM4ECIT
SCHEMBL8884848 0.79 XIAP (0.42)
SCHEMBL8882517 0.79 LNPEP (0.36) HTTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5620995-A Substituted heterocyclic carboxyamides, their preparation and their use as pharmaceuticals HOECHST AKTIENGESELLSCHAFT (DE) 1997-04-15 US disclosed