SCHEMBL8883802

SCHEMBL8883802

O=C(Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1)N1CC[C@@](CCN2CCN(C3CCCCC3)CC2)(c2ccc(Cl)c(Cl)c2)C1

nearest known ligand 0.53

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 11/20 0.53
TACR1 P25103 15/20 0.49
CCR5 P51681 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8883314 1.00 TACR2 (0.53) TACR2TACR1CCR5
SCHEMBL8883306 1.00 TACR2 (0.53) TACR2TACR1CCR5
SCHEMBL9027915 0.96 CCR5 (0.51) TACR2TACR1CCR5
SCHEMBL9027980 0.96 CCR5 (0.51) TACR2TACR1CCR5
SCHEMBL9027909 0.96 CCR5 (0.51) TACR2TACR1CCR5
SCHEMBL9028653 0.95 CCR5 (0.48) TACR2TACR1CCR5
SCHEMBL9027464 0.95 CCR5 (0.48) TACR2TACR1CCR5
SCHEMBL8884820 0.94 TACR2 (0.53) TACR2TACR1CCR5
SCHEMBL8884639 0.94 TACR2 (0.53) TACR2TACR1CCR5
SCHEMBL8884647 0.94 TACR2 (0.53) TACR2TACR1CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607947-A Pyrrolidinyl tachykinin receptor antagonists ELI LILLY AND COMPANY (US) 1997-03-04 US disclosed
EP-0714891-A1 Heterocyclic tachykinin receptor antagonists ELI LILLY AND COMPANY (US) 1996-06-05 EP disclosed