SCHEMBL8884639

SCHEMBL8884639

O=C(Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1)N1CC[C@](CCN2CCC(N3CCCCC3)CC2)(c2ccc(Cl)c(Cl)c2)C1

nearest known ligand 0.53

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 9/20 0.53
TACR1 P25103 13/20 0.50
CCR5 P51681 1/20 0.49
MCHR1 Q99705 3/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8884820 1.00 TACR2 (0.53) TACR2TACR1CCR5MCHR1
SCHEMBL8884647 1.00 TACR2 (0.53) TACR2TACR1CCR5MCHR1
SCHEMBL9028598 0.96 CCR5 (0.54) TACR2TACR1CCR5MCHR1
SCHEMBL9027461 0.96 CCR5 (0.54) TACR2TACR1CCR5MCHR1
SCHEMBL9028150 0.96 CCR5 (0.52) TACR2TACR1CCR5MCHR1
SCHEMBL9027473 0.96 CCR5 (0.54) TACR2TACR1CCR5MCHR1
SCHEMBL9028425 0.96 CCR5 (0.52) TACR2TACR1CCR5MCHR1
SCHEMBL8883802 0.94 TACR2 (0.53) TACR2TACR1CCR5
SCHEMBL8883306 0.94 TACR2 (0.53) TACR2TACR1CCR5
SCHEMBL8883314 0.94 TACR2 (0.53) TACR2TACR1CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607947-A Pyrrolidinyl tachykinin receptor antagonists ELI LILLY AND COMPANY (US) 1997-03-04 US disclosed
EP-0714891-A1 Heterocyclic tachykinin receptor antagonists ELI LILLY AND COMPANY (US) 1996-06-05 EP disclosed