SCHEMBL8884548

SCHEMBL8884548

CCOC(=O)CNC(=O)c1ccc2c(c1)C=CC(C)(C)O2

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.58
RAB9A P51151 3/20 0.58
TP53 P04637 1/20 0.58
GLA P06280 1/20 0.58
COXFA4 O00483 1/20 0.49
ALDH1A1 P00352 6/20 0.49
KDM4E B2RXH2 2/20 0.49
GAA P10253 1/20 0.49
SMN1; SMN2 Q16637 3/20 0.46
MAPT P10636 3/20 0.43
TDP1 Q9NUW8 2/20 0.41
POLB P06746 2/20 0.41
CYP3A4 P08684 1/20 0.41
HPGD P15428 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
BRCA1 P38398 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8884738 0.87 COXFA4 (0.48) NPC1RAB9ATP53GLACOXFA4
SCHEMBL8885682 0.82 NPC1 (0.58) NPC1RAB9ATP53GLAALDH1A1
SCHEMBL8883383 0.80 COXFA4 (0.52) NPC1RAB9ATP53COXFA4ALDH1A1
SCHEMBL8884505 0.80 COXFA4 (0.48) NPC1RAB9ATP53COXFA4ALDH1A1
SCHEMBL8885457 0.79 COXFA4 (0.47) NPC1RAB9ATP53COXFA4ALDH1A1
SCHEMBL8882853 0.75 NPC1 (0.56) NPC1RAB9ATP53ALDH1A1KDM4E
SCHEMBL11398330 0.75 COXFA4 (0.62) NPC1RAB9ATP53COXFA4ALDH1A1
SCHEMBL16865509 0.75 COXFA4 (0.56) NPC1RAB9ACOXFA4SMN1; SMN2
SCHEMBL16694306 0.74 HIF1A (0.62) COXFA4ALDH1A1SMN1; SMN2
SCHEMBL8885313 0.73 NPC1 (0.52) NPC1RAB9ACOXFA4ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5677324-A MUSCLE RELAXANTS PFIZER INC. (US) 1997-10-14 US disclosed
EP-0690855-B1 BENZOPYRANES AS POTASSIUM CHANNEL OPENERS PFIZER LTD (GB) 1996-12-18 EP disclosed
WO-1994020491-A1 BENZOPYRANES AS POTASSIUM CHANNEL OPENERS PFIZER LIMITED (GB) 1994-09-15 WO disclosed