SCHEMBL8884552

SCHEMBL8884552

CC(C)COc1ccnc(C(=O)NC(=O)CN)c1O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.36
TP53 P04637 3/20 0.36
NPC1 O15118 2/20 0.36
GAA P10253 2/20 0.36
HTT P42858 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
RAB9A P51151 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.34
SMPD1 P17405 2/20 0.33
POLB P06746 2/20 0.33
ALDH1A1 P00352 2/20 0.33
USP2 O75604 2/20 0.33
HPGD P15428 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
XDH P47989 1/20 0.32
EP300 Q09472 1/20 0.32
MEN1 O00255 1/20 0.32
ALOX15 P16050 1/20 0.32
TSHR P16473 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8881773 0.88 HTT (0.40) GAAHTTTDP1XDH
SCHEMBL8883058 0.86 GRIN3B (0.38) TP53TDP1
SCHEMBL8883715 0.86 SMN1; SMN2 (0.37) TP53NPC1GAASMN1; SMN2RAB9A
SCHEMBL8883971 0.85 CYP3A4 (0.35) MAPTTP53NPC1GAAHTT
SCHEMBL8884435 0.84 TDP1 (0.42) MAPTTP53NPC1HTTSMN1; SMN2
SCHEMBL8882459 0.84 IKBKB (0.39) MAPTNPC1GAAHTTSMN1; SMN2
SCHEMBL8883369 0.82 HPGD (0.37) NPC1GAAHTTSMN1; SMN2RAB9A
SCHEMBL8881872 0.82 SMN1; SMN2 (0.39) MAPTGAAHTTSMN1; SMN2SMPD1
SCHEMBL8882455 0.81 PTPN1 (0.41) MAPTNPC1SMN1; SMN2SMPD1MEN1
SCHEMBL8779122 0.81 MAPT (0.33) MAPTTP53NPC1GAAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5620995-A Substituted heterocyclic carboxyamides, their preparation and their use as pharmaceuticals HOECHST AKTIENGESELLSCHAFT (DE) 1997-04-15 US disclosed