SCHEMBL8884435

SCHEMBL8884435

COc1ccnc(C(=O)NC(=O)CN)c1O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.42
KLKB1 P03952 1/20 0.39
ATM Q13315 1/20 0.36
NPC1 O15118 3/20 0.35
CTSD P07339 1/20 0.35
LMNA P02545 2/20 0.34
CYP1A2 P05177 1/20 0.34
TSHR P16473 1/20 0.34
CYP2C19 P33261 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
ADRA1A P35348 1/20 0.34
GRIN3B O60391 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2C Q14957 1/20 0.34
TP53 P04637 2/20 0.34
KDM4E B2RXH2 2/20 0.34
IKBKB O14920 1/20 0.34
PKM P14618 1/20 0.34
RAB9A P51151 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8883715 0.88 SMN1; SMN2 (0.37) TDP1NPC1LMNAGRIN3BGRIN1
SCHEMBL8883369 0.87 HPGD (0.37) TDP1NPC1LMNAKDM4EIKBKB
SCHEMBL8883058 0.85 GRIN3B (0.38) TDP1LMNAGRIN3BGRIN1GRIN2C
SCHEMBL8882459 0.85 IKBKB (0.39) TDP1NPC1LMNATSHRCYP2C19
SCHEMBL8884552 0.84 MAPT (0.36) TDP1NPC1TSHRTP53RAB9A
SCHEMBL8881872 0.84 SMN1; SMN2 (0.39) LMNACYP1A2TSHRCYP2C19KDM4E
SCHEMBL8882455 0.83 PTPN1 (0.41) NPC1LMNACYP1A2CYP2C19MAPT
SCHEMBL8881773 0.82 HTT (0.40) TDP1KDM4EMAPK1HTT
SCHEMBL8882969 0.82 PTPN1 (0.43) NPC1LMNATSHRTP53MAPT
SCHEMBL8884367 0.82 CYP1A2 (0.40) CYP1A2KDM4EMAPTMAPK1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5620995-A Substituted heterocyclic carboxyamides, their preparation and their use as pharmaceuticals HOECHST AKTIENGESELLSCHAFT (DE) 1997-04-15 US disclosed