SCHEMBL88851

SCHEMBL88851

c1cc2nccnc2cn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4A O75164 1/20 0.39
KDM4B O94953 1/20 0.39
KDM5C P41229 1/20 0.39
KDM4C Q9H3R0 1/20 0.39
KDM5B Q9UGL1 1/20 0.39
KDM3A Q9Y4C1 1/20 0.39
MAPK1 P28482 1/20 0.39
HSP90AA1 P07900 1/20 0.38
FGFR1 P11362 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
ALDH1A1 P00352 3/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2A6 P11509 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
METAP2 P50579 1/20 0.33
METAP1 P53582 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29428806 1.00 KDM4A (0.39) KDM4AKDM4BKDM5CKDM4CKDM5B
SCHEMBL30237822 1.00 KDM4A (0.39) KDM4AKDM4BKDM5CKDM4CKDM5B
Pyrazine SCHEMBL7056616 0.95 HSP90AA1 (0.40) KDM4AKDM4BKDM5CKDM4CKDM5B
SCHEMBL14856779 0.82 ALDH1A1 (0.40) FGFR1NPC1RAB9AADORA3ALDH1A1
SCHEMBL5343673 0.76 KDM4C (0.40) KDM4AKDM4BKDM5CKDM4CKDM5B
SCHEMBL1263213 0.72 EGFR (0.33) KDM4AKDM4BKDM5CKDM4CKDM5B
SCHEMBL16878146 0.72 EGFR (0.33) KDM4AKDM4BKDM5CKDM4CKDM5B
SCHEMBL22479745 0.71 KDM4E (0.39) KDM4AKDM4BKDM5CKDM4CKDM5B
SCHEMBL21591641 0.71 ALDH1A1 (0.45) KDM4AKDM4BKDM5CKDM4CKDM5B
SCHEMBL22479748 0.71 ADORA3 (0.37) KDM4AKDM4BKDM5CKDM4CKDM5B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1263 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025076059-A1 ROCAGLATE DERIVATIVES AND USES THEREOF TRUSTEES OF BOSTON UNIVERSITY (US) 2025-04-10 WO claimed
US-12129381-B1 Single vessel solvent based method for making a Zn/Cu composite IMAM ABDULRAHMAN BIN FAISAL UNIVERSITY (SA) 2024-10-29 US claimed
US-20240336778-A1 SINGLE VESSEL SOLVENT BASED METHOD FOR MAKING A ZN/CU COMPOSITE IMAM ABDULRAHMAN BIN FAISAL UNIVERSITY (SA) 2024-10-10 US claimed
US-12031043-B2 Method for synthesizing a micro/nanosphere-containing composite IMAM ABDULRAHMAN BIN FAISAL UNIVERSITY (SA) 2024-07-09 US claimed
EP-4146222-A1 HETEROCYCLIC COMPOUNDS AS TRIGGERING RECEPTOR EXPRESSED ON MYELOID CELLS 2 AGONISTS AND METHODS OF USE Amgen Inc. (US) 2023-03-15 EP claimed
US-20230002617-A1 METHOD FOR SYNTHESIZING A MICRO/NANOSPHERE-CONTAINING COMPOSITE IMAM ABDULRAHMAN BIN FAISAL UNIVERSITY (SA) 2023-01-05 US claimed
US-11485862-B2 Metallophthalocyanine-ZnO hollow nanospheres composite IMAM ABDULRAHMAN BIN FAISAL UNIVERSITY (SA) 2022-11-01 US claimed
US-11111149-B2 Fly ash-catalyzed method for making graphene KING ABDULAZIZ UNIVERSITY (SA) 2021-09-07 US claimed
US-20210246029-A1 FLY ASH-CATALYZED METHOD FOR MAKING GRAPHENE KING ABDULAZIZ UNIVERSITY (SA) 2021-08-12 US claimed
US-11053125-B2 Graphene from fly ash KING ABDULAZIZ UNIVERSITY (SA) 2021-07-06 US claimed
US-RE37650-E1 Aryl and heteroaryl quinazoline compounds which inhibit CSF-1R receptor tyrosine kinase AVENTIS PHARMACETICAL PRODUCTS, INC. 2002-04-09 US claimed
CN-1320121-A Substituted 3-cyanoquinolines as protein tyrosine kinase inhibitors AMERICAN CYANAMID CO (US) 2001-10-31 CN claimed
US-6288082-B1 COMPOUNDS SUCH AS 6,7-DIETHOXY-4-(INDAN-5-YLAMINO) -QUINOLINE-3-CARBONITRILE USED AS ANTINEOPLASTIC AGENTS AND IN THE TREATMENT OF POLYCYCSTIC KIDNEY DISEASE AMERICAN CYANAMID COMPANY 2001-09-11 US claimed
EP-1117659-A1 SUBSTITUTED 3-CYANOQUINOLINES AS PROTEIN TYROSINE KINASES INHIBITORS American Cyanamid Company (US) 2001-07-25 EP claimed
WO-2000018761-A1 SUBSTITUTED 3-CYANOQUINOLINES AS PROTEIN TYROSINE KINASES INHIBITORS AMERICAN CYANAMID COMPANY (US) 2000-04-06 WO claimed
EP-0145337-B1 ELECTROCHROMIC DEVICES CHEVRON RESEARCH AND TECHNOLOGY COMPANY (US) 1990-08-08 EP claimed
EP-0096723-B1 BATTERIES FABRICATED WITH ELECTROACTIVE POLYMERS CHEVRON RESEARCH AND TECHNOLOGY COMPANY (US) 1988-08-10 EP claimed
US-4613211-A REVERSE COLOR CHANGING POLYMER FILM AS DISPLAY ELECTRODE CHEVRON RESEARCH COMPANY (US) 1986-09-23 US claimed
US-4579679-A Electroactive polymers CHEVRON RESEARCH COMPANY (US) 1986-04-01 US claimed
EP-0145337-A2 Electrochromic devices CHEVRON RESEARCH AND TECHNOLOGY COMPANY (US) 1985-06-19 EP claimed