SCHEMBL8885256

SCHEMBL8885256

c1cnc(NCCCNCC2CCc3cnccc3O2)nc1

nearest known ligand 0.78

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 18/20 0.78
HTR1D P28221 18/20 0.78
ADRA1D P25100 1/20 0.48
ADRA1A P35348 1/20 0.48
ADRA1B P35368 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8864158 0.85 HTR1A (0.95) HTR1AHTR1DADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL8864153 0.85 HTR1A (0.95) HTR1AHTR1DADRA1DADRA1AADRA1B
SCHEMBL8880289 0.83 HTR1A (0.74) HTR1AHTR1D
SCHEMBL8863907 0.81 HTR1A (0.72) HTR1AHTR1D
SCHEMBL8885185 0.81 HTR1A (0.75) HTR1AHTR1DADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL8887313 0.80 HTR1A (0.73) HTR1AHTR1DADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL9051868 0.79 HTR1A (0.69) HTR1AHTR1DADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL9051866 0.79 HTR1A (0.69) HTR1AHTR1DADRA1DADRA1AADRA1B
Oxalic Acid SCHEMBL8864004 0.79 HTR1A (0.68) HTR1AHTR1D
Oxalic Acid SCHEMBL8864011 0.79 HTR1A (0.68) HTR1AHTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691344-A Vasoconstrictive substituted dihydropyranopyridines JANSSEN PHARMACEUTICA, N.V. (BE) 1997-11-25 US claimed
EP-0714395-A1 VASOCONSTRICTIVE SUBSTITUTED DIHYDROPYRANOPYRIDINES JANSSEN PHARMACEUTICA N.V. (BE) 1996-06-05 EP claimed
WO-1995005381-A1 VASOCONSTRICTIVE SUBSTITUTED DIHYDROPYRANOPYRIDINES JANSSEN PHARMACEUTICA N.V. (BE) 1995-02-23 WO claimed
US-5691344-A Vasoconstrictive substituted dihydropyranopyridines JANSSEN PHARMACEUTICA, N.V. (BE) 1997-11-25 US disclosed
EP-0714395-A1 VASOCONSTRICTIVE SUBSTITUTED DIHYDROPYRANOPYRIDINES JANSSEN PHARMACEUTICA N.V. (BE) 1996-06-05 EP disclosed
WO-1995005381-A1 VASOCONSTRICTIVE SUBSTITUTED DIHYDROPYRANOPYRIDINES JANSSEN PHARMACEUTICA N.V. (BE) 1995-02-23 WO disclosed