SCHEMBL8885484

SCHEMBL8885484

CN(C)Cc1cc(CO)co1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.34
KDM4E B2RXH2 2/20 0.34
GAA P10253 2/20 0.34
MEN1 O00255 1/20 0.34
POLB P06746 1/20 0.34
MAPT P10636 1/20 0.34
THRB P10828 1/20 0.34
G6PD P11413 1/20 0.34
PABPC1 P11940 1/20 0.34
KMT2A Q03164 1/20 0.34
HKDC1 Q2TB90 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
TYR P14679 1/20 0.34
DAO P14920 1/20 0.34
ACHE P22303 4/20 0.33
BCHE P06276 2/20 0.33
ALOX15 P16050 2/20 0.32
TSHR P16473 2/20 0.32
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9034411 0.84 KDM4E (0.42) ALDH1A1KDM4EGAAMEN1POLB
SCHEMBL901473 0.78
SCHEMBL10175116 0.77
SCHEMBL8132166 0.70 SLC6A2 (0.54) ALDH1A1MEN1MAPTKMT2ACYP2C19
SCHEMBL19331285 0.69 TYR (0.63) KDM4ETYRDAO
SCHEMBL1876155 0.69 ALDH1A1 (0.48) ALDH1A1KDM4EGAAMEN1POLB
SCHEMBL11389129 0.68 NPC1 (0.46) ALDH1A1GAAMAPTKMT2ADAO
SCHEMBL2735671 0.67
SCHEMBL11171888 0.67 CYP1A2 (0.44) ALDH1A1MEN1MAPTKMT2ADAO
SCHEMBL358651 0.67 IDH1 (0.57) MEN1KMT2ATDP1DAOALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5661146-A ANALGESICS G.D. SEARLE & CO. (US) 1997-08-26 US disclosed
US-5504077-A ANALGESICS G. D. SEARLE & CO. (US) 1996-04-02 US disclosed
WO-1995033733-A1 SUBSTITUTED DIBENZOXAZEPINE AND DIBENZOTHIAZEPINE UREAS USEFUL AS PROSTAGLANDIN ANTAGONISTS G.D. SEARLE & CO. (US) 1995-12-14 WO disclosed
WO-1995033734-A1 SUBSTITUTED DIBENZOXAZEPINE AND DIBENZTHIAZEPINE CARBAMATES USEFUL AS PROSTAGLANDIN ANTAGONISTS G.D. SEARLE & CO. (US) 1995-12-14 WO disclosed
US-5449675-A Analgesics G. D. SEARLE & CO. (US) 1995-09-12 US disclosed
US-5441950-A Analgesics, prostaglandin E2 antagonists G. D. SEARLE & CO. (US) 1995-08-15 US disclosed