SCHEMBL8886779

SCHEMBL8886779

CCCNC1CNc2ccccc2C1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.52
EPHX2 P34913 1/20 0.50
DRD2 P14416 7/20 0.46
DRD3 P35462 6/20 0.46
DRD4 P21917 3/20 0.46
MTNR1A P48039 1/20 0.46
MTNR1B P49286 1/20 0.46
HTR1A P08908 3/20 0.43
GRIN2B Q13224 2/20 0.41
HTR1D P28221 1/20 0.40
HTR1B P28222 1/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5898226 1.00 SIGMAR1 (0.52) SIGMAR1EPHX2DRD2DRD3DRD4
Hydrochloric Acid SCHEMBL4796338 0.98 SIGMAR1 (0.51) SIGMAR1EPHX2DRD2DRD3DRD4
SCHEMBL11213075 0.90 EPHX2 (0.47) SIGMAR1EPHX2DRD2DRD3DRD4
SCHEMBL1792787 0.79 GRIN2B (0.61) SIGMAR1DRD2DRD3DRD4MTNR1A
SCHEMBL4798922 0.78 EPHX2 (0.56) SIGMAR1EPHX2DRD2DRD3DRD4
SCHEMBL4798460 0.78 EPHX2 (0.56) SIGMAR1EPHX2DRD2DRD3DRD4
SCHEMBL9675361 0.76 DRD2 (0.44) SIGMAR1DRD2DRD3DRD4HTR1A
SCHEMBL8569808 0.75 EPHX2 (0.64) EPHX2MTNR1AMTNR1B
SCHEMBL8569805 0.75 EPHX2 (0.64) EPHX2MTNR1AMTNR1B
SCHEMBL8569806 0.75 EPHX2 (0.64) EPHX2MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5650427-A ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1997-07-22 US disclosed
US-5461061-A Antidepressants WIKSTROM HAKAN V (NL) 1995-10-24 US disclosed
US-5288748-A Antidepressants THE UPJOHN COMPANY (US) 1994-02-22 US disclosed
EP-0510068-A1 NEW CENTRALLY ACTING 6,7,8,9-TETRAHYDRO-3H-BENZ(e)INDOLE HETEROCYCLICS PHARMACIA & UPJOHN COMPANY (US) 1992-10-28 EP disclosed
WO-1991011435-A2 NEW CENTRALLY ACTING 6,7,8,9-TETRAHYDRO-3H-BENZ(e)INDOLE HETEROCYCLICS THE UPJOHN COMPANY (US) 1991-08-08 WO disclosed