SCHEMBL8887102

SCHEMBL8887102

CCn1nc(-c2ccccc2)c(-c2ccc(=O)n(C)n2)c1-c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 3/20 0.46
PDE4B Q07343 3/20 0.46
PDE4C Q08493 3/20 0.46
PDE4D Q08499 3/20 0.46
SMN1; SMN2 Q16637 1/20 0.44
PTGIR P43119 1/20 0.43
BRD4 O60885 2/20 0.43
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
USP2 O75604 1/20 0.42
TNNI3 P19429 1/20 0.42
CRHBP P24387 1/20 0.42
MAPK1 P28482 1/20 0.42
CASP1 P29466 1/20 0.42
TNNT2 P45379 1/20 0.42
CASP7 P55210 1/20 0.42
TNNC1 P63316 1/20 0.42
KMT2A Q03164 1/20 0.42
ATM Q13315 1/20 0.42
CRHR2 Q13324 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8888600 0.86 KDM4E (0.41) PDE4APDE4BPDE4CPDE4DSMN1; SMN2
SCHEMBL8889113 0.79 CYP1A2 (0.50) PDE4APDE4BPDE4CPDE4DSMN1; SMN2
SCHEMBL11142730 0.74 KMT2A (0.53) SMN1; SMN2BRD4KDM4EMEN1KMT2A
SCHEMBL8809138 0.73 ADORA1 (0.64) BRD4MAPK1ADORA1ADORA3
SCHEMBL7373031 0.72 ADORA1 (0.48) BRD4MAPK1KMT2AADORA1ADORA3
SCHEMBL11397967 0.71 HRH3 (0.54) SMN1; SMN2BRD4KDM4EMEN1KMT2A
SCHEMBL27659542 0.71 BRD4 (0.47) SMN1; SMN2BRD4KDM4EMEN1KMT2A
SCHEMBL11862067 0.70 CA1 (0.56) PDE4APDE4BPDE4CPDE4DSMN1; SMN2
SCHEMBL4054492 0.70 HTT (0.62) SMN1; SMN2KDM4EMEN1KMT2ATP53
SCHEMBL8889100 0.69 PTGIR (0.49) PDE4APDE4BPDE4CPDE4DPTGIR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997001551-A1 PYRAZOLE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-01-16 WO disclosed