SCHEMBL8889113

SCHEMBL8889113

CCn1nc(-c2ccccc2)c(-c2ccc(=O)[nH]n2)c1-c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.50
PDE4A P27815 4/20 0.47
PDE4B Q07343 4/20 0.47
PDE4C Q08493 4/20 0.47
PDE4D Q08499 4/20 0.47
SMN1; SMN2 Q16637 1/20 0.43
PDE5A O76074 1/20 0.42
PDE3A Q14432 1/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
KDM4E B2RXH2 1/20 0.41
USP2 O75604 1/20 0.41
TNNI3 P19429 1/20 0.41
CRHBP P24387 1/20 0.41
MAPK1 P28482 1/20 0.41
CASP1 P29466 1/20 0.41
TNNT2 P45379 1/20 0.41
CASP7 P55210 1/20 0.41
TNNC1 P63316 1/20 0.41
ATM Q13315 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8889100 0.87 PTGIR (0.49) CYP1A2PDE4APDE4BPDE4CPDE4D
SCHEMBL8887697 0.87 CYP1A2 (0.47) CYP1A2PDE4APDE4BPDE4CPDE4D
SCHEMBL8889588 0.86 CYP1A2 (0.49) CYP1A2PDE4APDE4BPDE4CPDE4D
SCHEMBL8890203 0.84 CYP1A2 (0.47) CYP1A2PDE4APDE4BPDE4CPDE4D
SCHEMBL8888651 0.84 CYP1A2 (0.55) CYP1A2SMN1; SMN2PDE5APDE3AMEN1
SCHEMBL8887601 0.81 LMNA (0.48) CYP1A2PDE4APDE4BPDE4CPDE4D
SCHEMBL8887102 0.79 PDE4A (0.46) PDE4APDE4BPDE4CPDE4DSMN1; SMN2
SCHEMBL8889716 0.78 PDE4A (0.52) CYP1A2PDE4APDE4BPDE4CPDE4D
SCHEMBL5807524 0.76 CYP1A2 (0.51) CYP1A2SMN1; SMN2PDE5APDE3AMEN1
Bromide SCHEMBL5806494 0.72 CYP1A2 (0.50) CYP1A2PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997001551-A1 PYRAZOLE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-01-16 WO disclosed