SCHEMBL8887549

SCHEMBL8887549

c1ccc(C(c2ccccc2)(c2ccccc2)c2cc[nH]n2)cc1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 2/20 0.33
MAPK1 P28482 1/20 0.33
TSHR P16473 3/20 0.32
ALDH1A1 P00352 2/20 0.32
ALOX15 P16050 1/20 0.31
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27733507 0.89 ALDH1A1 (0.33) MAPK1ALDH1A1
SCHEMBL20772230 0.89 KIF11 (0.31)
SCHEMBL8123393 0.85 ALDH1A1 (0.39) ALDH1A1
SCHEMBL2766738 0.79 ALDH1A1 (0.41) KCNN4MAPK1TSHRALDH1A1ALOX15
SCHEMBL13221175 0.79 ESR1 (0.41) KCNN4MAPK1TSHRALDH1A1ALOX15
SCHEMBL7218962 0.79 KCNN4 (0.34) KCNN4MAPK1TSHRALDH1A1
SCHEMBL25373363 0.77
SCHEMBL11143506 0.76 ATM (0.33)
SCHEMBL29196149 0.75 MAPT (0.34) MAPK1TSHRALDH1A1HPGD
SCHEMBL11501301 0.74 CYP2C9 (0.46) KCNN4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105050598-B Novel compounds as ERK inhibitors 默沙东公司 2018-04-27 CN disclosed
WO-1997001551-A1 PYRAZOLE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-01-16 WO disclosed
CN-1116425-A New cephem compounds FUJISAWA PHARMACEUTICAL CO (JP) 1996-02-07 CN disclosed
EP-0091130-B1 CEPHALOSPORIN DERIVATIVES, PROCESS FOR PREPARING AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAID COMPOUNDS DAIICHI SEIYAKU CO., LTD. (JP) 1987-04-08 EP disclosed