SCHEMBL8887771

SCHEMBL8887771

CCOC(=O)CSCc1cc(C(=O)OC)ccc1NC(C)=O

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.48
ALDH1A1 P00352 7/20 0.47
HPGD P15428 2/20 0.44
MAPT P10636 5/20 0.44
SMN1; SMN2 Q16637 4/20 0.44
HSD17B10 Q99714 2/20 0.44
NPC1 O15118 4/20 0.42
KDM4E B2RXH2 4/20 0.41
LMNA P02545 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
MEN1 O00255 1/20 0.41
RAB9A P51151 4/20 0.40
STAT1 P42224 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8888198 0.85 KMT2A (0.52) KMT2AALDH1A1HPGDMAPTSMN1; SMN2
SCHEMBL8887242 0.76 ALDH1A1 (0.59) KMT2AALDH1A1HPGDSMN1; SMN2HSD17B10
SCHEMBL11623111 0.75 ALDH1A1 (0.57) KMT2AALDH1A1HPGDMAPTSMN1; SMN2
SCHEMBL5682853 0.75 KMT2A (0.61) KMT2AALDH1A1HPGDMAPTSMN1; SMN2
SCHEMBL11622464 0.75 ALDH1A1 (0.54) KMT2AALDH1A1HPGDMAPTSMN1; SMN2
SCHEMBL8888165 0.74 ALDH1A1 (0.56) KMT2AALDH1A1HPGDMAPTSMN1; SMN2
SCHEMBL8886566 0.74 ALDH1A1 (0.56) KMT2AALDH1A1HPGDSMN1; SMN2HSD17B10
SCHEMBL18394312 0.73 ALDH1A1 (0.49) KMT2AALDH1A1HPGDMAPTSMN1; SMN2
SCHEMBL19068409 0.73 ALDH1A1 (0.55) KMT2AALDH1A1HPGDMAPTSMN1; SMN2
SCHEMBL5686135 0.73 KMT2A (0.58) KMT2AALDH1A1MAPTSMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5602277-A Substituted benzene derivatives useful as neuraminidase inhibitors BIOCRYST PHARMACEUTICALS, INC. (US) 1997-02-11 US disclosed
WO-1996030329-A1 SUBSTITUTED BENZENE DERIVATIVES USEFUL AS NEURAMINIDASE INHIBITORS BIOCRYST PHARMACEUTICALS, INCORPORATED (US) 1996-10-03 WO disclosed