SCHEMBL8889178

SCHEMBL8889178

Cc1nn(COCC[Si](C)(C)C)c2cc(Br)c(Br)cc12

nearest known ligand 0.41

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 4/20 0.41
ADORA2B P29275 4/20 0.41
DGAT1 O75907 3/20 0.36
NPC1 O15118 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8226285 0.90 DGAT1 (0.40) ADORA2AADORA2BDGAT1NPC1
SCHEMBL4312796 0.84 DGAT1 (0.43) ADORA2AADORA2BDGAT1NPC1
SCHEMBL11976878 0.84 DGAT1 (0.43) ADORA2AADORA2BDGAT1NPC1
SCHEMBL14493341 0.81 ADORA2A (0.37) ADORA2AADORA2BDGAT1NPC1
SCHEMBL23533512 0.79 DGAT1 (0.34) DGAT1NPC1
SCHEMBL30284929 0.78 ADORA2A (0.36) ADORA2AADORA2BDGAT1NPC1
SCHEMBL29612533 0.78 NPC1 (0.38) ADORA2AADORA2BDGAT1NPC1
SCHEMBL2144240 0.78 ADORA2A (0.36) ADORA2AADORA2BDGAT1NPC1
SCHEMBL19023399 0.78 NPC1 (0.38) ADORA2AADORA2BDGAT1NPC1
SCHEMBL26039082 0.77 DGAT1 (0.38) ADORA2AADORA2BDGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5631264-A NEUROLOGICAL DISORDERS SANOFI WINTHROP, INC. (US) 1997-05-20 US disclosed
US-5554620-A Substituted 6,11-ethano-6,11-dihydrobenzo[b] quinolizinium salts and compositions and methods of use thereof STERLING WINTHROP INC. (US) 1996-09-10 US disclosed