SCHEMBL8889395

SCHEMBL8889395

COc1ccc(C(=O)Nc2c(Cl)cncc2Cl)cc1-c1ccc2ccccc2c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 11/20 0.65
PDE4B Q07343 10/20 0.55
PDE4A P27815 9/20 0.55
PDE4C Q08493 9/20 0.55
CYP2B6 P20813 1/20 0.54
NPC1 O15118 1/20 0.50
NQO2 P16083 1/20 0.50
CASP3 P42574 1/20 0.50
RAB9A P51151 1/20 0.50
SENP7 Q9BQF6 1/20 0.50
HSP90AA1 P07900 1/20 0.49
HSP90AB1 P08238 1/20 0.49
SIRT2 Q8IXJ6 1/20 0.49
PDE3B Q13370 1/20 0.47
PDE11A Q9HCR9 1/20 0.47
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
KMT2A Q03164 1/20 0.47
HPSE Q9Y251 2/20 0.47
ABL1 P00519 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8890532 0.87 PDE4D (0.70) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL8890076 0.84 PDE4D (0.66) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL8889523 0.81 PDE4D (0.61) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL8900612 0.80 PDE4D (0.60) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL8889534 0.80 PDE4D (0.60) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL8890316 0.80 PDE4D (0.66) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL15270505 0.79 PDE4D (1.00) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL8898765 0.78 ALOX15 (0.65) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL8890618 0.78 PDE4D (0.66) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL2908650 0.77 PDE4D (0.81) PDE4DPDE4BPDE4APDE4CCYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997003967-A1 SUBSTITUTED AROMATIC COMPOUNDS AND THEIR PHARMACEUTICAL USE RHONE-POULENC RORER LIMITED (GB) 1997-02-06 WO claimed
WO-1997003967-A1 SUBSTITUTED AROMATIC COMPOUNDS AND THEIR PHARMACEUTICAL USE RHONE-POULENC RORER LIMITED (GB) 1997-02-06 WO disclosed