SCHEMBL8890243

SCHEMBL8890243

COc1ccc(C(=O)O)cc1-c1nc(-c2ccccn2)no1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 10/20 0.68
RAB9A P51151 9/20 0.68
SMN1; SMN2 Q16637 9/20 0.68
PKM P14618 8/20 0.68
TP53 P04637 7/20 0.68
HSD17B10 Q99714 4/20 0.68
KDM4E B2RXH2 3/20 0.68
GAA P10253 2/20 0.68
MAPT P10636 5/20 0.60
ALDH1A1 P00352 4/20 0.60
GRM5 P41594 4/20 0.53
L3MBTL1 Q9Y468 3/20 0.52
MITF O75030 1/20 0.52
HSP90AA1 P07900 1/20 0.52
POLB P06746 1/20 0.51
S1PR1 P21453 1/20 0.50
KMT2A Q03164 1/20 0.50
TSHR P16473 3/20 0.49
MAPK1 P28482 2/20 0.49
HPGD P15428 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8890122 0.90 NPC1 (0.67) NPC1RAB9ASMN1; SMN2PKMTP53
SCHEMBL8898716 0.84 NPC1 (0.60) NPC1RAB9ASMN1; SMN2TP53HSD17B10
SCHEMBL13117741 0.84 KDM4C (0.60) RAB9AKDM4EMAPTKMT2ATSHR
SCHEMBL4345197 0.83 NPC1 (0.74) NPC1RAB9ASMN1; SMN2PKMTP53
SCHEMBL6451282 0.83 NPC1 (0.74) NPC1RAB9ASMN1; SMN2PKMTP53
SCHEMBL4197833 0.82 NPC1 (0.73) NPC1RAB9ASMN1; SMN2PKMTP53
SCHEMBL4183752 0.82 NPC1 (0.73) NPC1RAB9ASMN1; SMN2PKMTP53
SCHEMBL27572517 0.81 NPC1 (1.00) NPC1RAB9ASMN1; SMN2PKMTP53
SCHEMBL8890415 0.81 PDE4D (0.56) NPC1RAB9ASMN1; SMN2PKMTP53
SCHEMBL8890246 0.81 POLB (0.61) NPC1RAB9ASMN1; SMN2PKMTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997003967-A1 SUBSTITUTED AROMATIC COMPOUNDS AND THEIR PHARMACEUTICAL USE RHONE-POULENC RORER LIMITED (GB) 1997-02-06 WO disclosed