SCHEMBL8890415

SCHEMBL8890415

COc1ccc(C(=O)Nc2c(Cl)cncc2Cl)cc1-c1nc(-c2ccccn2)no1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 8/20 0.56
NPC1 O15118 3/20 0.54
HSD17B10 Q99714 2/20 0.54
TP53 P04637 2/20 0.54
RAB9A P51151 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
KDM4E B2RXH2 1/20 0.54
GAA P10253 1/20 0.54
PKM P14618 1/20 0.54
PDE4A P27815 6/20 0.51
PDE4B Q07343 6/20 0.51
PDE4C Q08493 6/20 0.51
CYP2B6 P20813 1/20 0.50
ALOX15 P16050 1/20 0.49
CASP1 P29466 1/20 0.49
CASP7 P55210 1/20 0.49
ALDH1A1 P00352 4/20 0.48
MAPT P10636 2/20 0.48
GRM5 P41594 4/20 0.47
ADORA3 P0DMS8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8900612 0.87 PDE4D (0.60) PDE4DNPC1HSD17B10TP53RAB9A
SCHEMBL8890668 0.84 PDE4D (0.57) PDE4DNPC1HSD17B10TP53RAB9A
SCHEMBL8898765 0.83 ALOX15 (0.65) PDE4DNPC1HSD17B10TP53RAB9A
SCHEMBL8890122 0.82 NPC1 (0.67) NPC1HSD17B10TP53RAB9ASMN1; SMN2
SCHEMBL8890243 0.81 NPC1 (0.68) NPC1HSD17B10TP53RAB9ASMN1; SMN2
SCHEMBL4183752 0.77 NPC1 (0.73) NPC1HSD17B10TP53RAB9ASMN1; SMN2
SCHEMBL4192484 0.76 NPC1 (0.60) NPC1HSD17B10TP53RAB9ASMN1; SMN2
SCHEMBL8890076 0.76 PDE4D (0.66) PDE4DPDE4APDE4BPDE4CCYP2B6
SCHEMBL8891692 0.76 PDE4D (0.52) PDE4DNPC1TP53RAB9ASMN1; SMN2
SCHEMBL8889395 0.75 PDE4D (0.65) PDE4DNPC1RAB9APDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997003967-A1 SUBSTITUTED AROMATIC COMPOUNDS AND THEIR PHARMACEUTICAL USE RHONE-POULENC RORER LIMITED (GB) 1997-02-06 WO claimed