SCHEMBL8890400

SCHEMBL8890400

Nc1cccc(CC2COc3ccc(O)cc3C2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTB4R Q15722 1/20 0.41
LTB4R2 Q9NPC1 1/20 0.41
HDAC1 Q13547 1/20 0.40
CYP19A1 P11511 4/20 0.39
CYP11B2 P19099 1/20 0.39
SIGMAR1 Q99720 2/20 0.39
HTR1A P08908 1/20 0.39
ESR1 P03372 1/20 0.39
ESR2 Q92731 1/20 0.39
DRD3 P35462 2/20 0.37
ALOX5 P09917 1/20 0.36
DRD2 P14416 1/20 0.36
DRD4 P21917 1/20 0.36
CA12 O43570 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9221077 0.82 LTB4R (0.46) LTB4RLTB4R2HDAC1CYP19A1SIGMAR1
SCHEMBL8888420 0.78 MTNR1A (0.44) LTB4RLTB4R2HDAC1MTNR1A
SCHEMBL28330990 0.74 CHRM5 (0.41) LTB4RLTB4R2CYP19A1CA1CA2
SCHEMBL28332417 0.74 CHRM5 (0.41) LTB4RLTB4R2CYP19A1CA1CA2
SCHEMBL8891775 0.74 LTB4R (0.41) LTB4R
SCHEMBL8888895 0.74 LTB4R (0.53) LTB4RLTB4R2CYP19A1
SCHEMBL22369104 0.73 MAOB (0.46) CYP19A1CYP11B2SIGMAR1CA1CA2
SCHEMBL28101525 0.70 ESR1 (0.47) HTR1AESR1ESR2DRD3DRD2
SCHEMBL28330978 0.69 CYP19A1 (0.57) LTB4RLTB4R2CYP19A1ESR1ESR2
SCHEMBL24228739 0.69 DRD3 (0.46) ESR1ESR2DRD3DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5641789-A INHIBITORS OF LEUKOTRIENES AND/OR BLOCKERS OF LEUKOTRIENE RECEPTORS; USEFUL IN PREVENTION OR TREATMENT OF ASTHMA, ARTHRITIS, PSORIASIS, ULCERS, MYOCARDIAL INFARCTION PFIZER INC. (US) 1997-06-24 US disclosed
CN-1090282-A The cycloalkyl that benzenefused, hydroxy replaces and the sulfone amide derivative of heterogeneous ring compound PFIZER (US) 1994-08-03 CN disclosed