SCHEMBL8890403

SCHEMBL8890403

COC(=O)c1ccc(OC)c(OCc2ccccn2)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 8/20 0.57
AURKB Q96GD4 2/20 0.57
INCENP Q9NQS7 2/20 0.57
MAPT P10636 2/20 0.54
HDAC1 Q13547 2/20 0.53
SMPD1 P17405 1/20 0.53
HDAC8 Q9BY41 1/20 0.53
HDAC6 Q9UBN7 1/20 0.53
PARP10 Q53GL7 1/20 0.52
MEN1 O00255 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP2C19 P33261 1/20 0.52
KMT2A Q03164 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
KDM4E B2RXH2 2/20 0.52
MTNR1A P48039 1/20 0.51
MTNR1B P49286 1/20 0.51
HDAC2 Q92769 1/20 0.51
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8891047 0.89 SYK (0.62) SYKAURKBINCENPMAPTHDAC1
SCHEMBL8892307 0.89 KDM4E (0.52) SYKAURKBINCENPMAPTMEN1
SCHEMBL4319936 0.87 SYK (0.56) SYKAURKBINCENPMAPTHDAC1
SCHEMBL31691389 0.83 KMT2A (0.47) SYKAURKBINCENPMAPTMEN1
SCHEMBL2188210 0.82 SMPD1 (0.76) MAPTHDAC1SMPD1HDAC8HDAC6
SCHEMBL17835555 0.81 MAPT (0.57) SYKMAPTMEN1CYP1A2CYP2C19
SCHEMBL30320388 0.81 PARP10 (0.69) SYKAURKBINCENPMAPTPARP10
SCHEMBL1732629 0.81 PARP10 (0.69) SYKAURKBINCENPMAPTPARP10
SCHEMBL8891644 0.80 MAPT (0.60) MAPTHDAC1SMPD1HDAC8HDAC6
SCHEMBL8890013 0.80 KDM4E (0.61) SYKAURKBINCENPMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997003967-A1 SUBSTITUTED AROMATIC COMPOUNDS AND THEIR PHARMACEUTICAL USE RHONE-POULENC RORER LIMITED (GB) 1997-02-06 WO disclosed