SCHEMBL8891047

SCHEMBL8891047

COc1ccc(C(=O)O)cc1OCc1ccccn1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 7/20 0.62
AURKB Q96GD4 2/20 0.62
INCENP Q9NQS7 2/20 0.62
KDM4E B2RXH2 1/20 0.60
MAPT P10636 1/20 0.60
CA12 O43570 1/20 0.59
CA1 P00915 1/20 0.59
CA2 P00918 1/20 0.59
CA4 P22748 1/20 0.59
CA6 P23280 1/20 0.59
CA7 P43166 1/20 0.59
TPMT P51580 1/20 0.59
CA9 Q16790 1/20 0.59
CA14 Q9ULX7 1/20 0.59
RXRA P19793 1/20 0.56
MRGPRX4 Q96LA9 3/20 0.56
SMPD1 P17405 1/20 0.55
HDAC1 Q13547 1/20 0.55
HDAC8 Q9BY41 1/20 0.55
HDAC6 Q9UBN7 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8890013 0.90 KDM4E (0.61) SYKAURKBINCENPKDM4EMAPT
SCHEMBL8890403 0.89 SYK (0.57) SYKAURKBINCENPKDM4EMAPT
SCHEMBL17844308 0.84 KDM4E (0.61) SYKAURKBINCENPKDM4EMAPT
SCHEMBL17810923 0.84 NPC1 (0.53) SYKAURKBINCENPKDM4EMAPT
SCHEMBL17810925 0.84 NPC1 (0.53) SYKAURKBINCENPKDM4EMAPT
SCHEMBL29375753 0.84 SMPD1 (0.75) KDM4ECA12CA1CA2CA4
SCHEMBL1029034 0.84 SMPD1 (0.75) KDM4ECA12CA1CA2CA4
SCHEMBL31691456 0.84 KDM4E (0.55) SYKAURKBINCENPKDM4EMAPT
SCHEMBL4314016 0.83 SYK (0.58) SYKAURKBINCENPKDM4EMAPT
SCHEMBL11271923 0.83 SMPD1 (0.73) KDM4ECA12CA1CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997003967-A1 SUBSTITUTED AROMATIC COMPOUNDS AND THEIR PHARMACEUTICAL USE RHONE-POULENC RORER LIMITED (GB) 1997-02-06 WO disclosed