SCHEMBL8890463

SCHEMBL8890463

CCOC(=O)c1ccc(NC(=O)C(C)C)c([N+](=O)[O-])c1

nearest known ligand 0.76

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.76
ALDH1A1 P00352 5/20 0.67
MAPT P10636 5/20 0.67
RAB9A P51151 3/20 0.67
NPC1 O15118 2/20 0.67
PKM P14618 1/20 0.67
CRHBP P24387 1/20 0.67
CRHR2 Q13324 1/20 0.67
LMNA P02545 2/20 0.65
KDM4E B2RXH2 1/20 0.65
POLB P06746 1/20 0.65
PTGER4 P35408 1/20 0.63
SMN1; SMN2 Q16637 2/20 0.53
HCAR3 P49019 1/20 0.51
TDP1 Q9NUW8 1/20 0.50
GAA P10253 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6170744 0.86 KMT2A (1.00) KMT2AALDH1A1MAPTRAB9ANPC1
SCHEMBL4332105 0.85 KMT2A (0.71) KMT2AALDH1A1MAPTRAB9ANPC1
SCHEMBL11609033 0.85 KMT2A (0.64) KMT2AALDH1A1MAPTRAB9ANPC1
SCHEMBL1965205 0.83 KMT2A (0.76) KMT2AALDH1A1MAPTRAB9ANPC1
SCHEMBL22382354 0.82 MAPT (0.81) KMT2AALDH1A1MAPTRAB9ANPC1
SCHEMBL31424609 0.82 KMT2A (0.67) KMT2AALDH1A1MAPTRAB9ANPC1
SCHEMBL15618391 0.81 HCAR3 (0.73) KMT2AALDH1A1MAPTRAB9ANPC1
SCHEMBL9043092 0.81 KMT2A (0.72) KMT2AALDH1A1MAPTRAB9ANPC1
SCHEMBL753425 0.81 KMT2A (0.72) KMT2AALDH1A1MAPTRAB9ANPC1
SCHEMBL6170341 0.81 KMT2A (0.59) KMT2AALDH1A1MAPTRAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5602277-A Substituted benzene derivatives useful as neuraminidase inhibitors BIOCRYST PHARMACEUTICALS, INC. (US) 1997-02-11 US disclosed
WO-1996030329-A1 SUBSTITUTED BENZENE DERIVATIVES USEFUL AS NEURAMINIDASE INHIBITORS BIOCRYST PHARMACEUTICALS, INCORPORATED (US) 1996-10-03 WO disclosed