SCHEMBL8890559

SCHEMBL8890559

COCCON(c1ccccc1)c1nc(Nc2ccc(Cl)cc2)c2cccc(OC(C)=O)c2n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 3/20 0.38
MAPT P10636 2/20 0.38
TP53 P04637 1/20 0.38
ROCK2 O75116 1/20 0.37
NPY5R Q15761 4/20 0.36
ALK Q9UM73 1/20 0.35
EGFR P00533 1/20 0.35
PDE5A O76074 2/20 0.35
ABCG2 Q9UNQ0 2/20 0.35
ABCC1 P33527 1/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
HPGD P15428 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
LMNA P02545 1/20 0.34
PIM1 P11309 1/20 0.34
PIM2 Q9P1W9 1/20 0.34
KDM1A O60341 1/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8891547 0.83 KDM1A (0.42) MAPTTP53NPY5RALKPDE5A
Hydrochloric Acid SCHEMBL8920462 0.82 KDM1A (0.42) MAPTTP53NPY5RALKALDH1A1
SCHEMBL8898287 0.66 HTR2A (0.41) KDRMAPTTP53NPY5RALK
SCHEMBL8890323 0.66 NPY5R (0.45) KDRNPY5REGFR
SCHEMBL8898291 0.66 CCR4 (0.38) NPY5R
Hydrochloric Acid SCHEMBL8890553 0.65 NPY5R (0.44) NPY5REGFR
Hydrochloric Acid SCHEMBL8892373 0.64 EGFR (0.49) KDREGFRKDM4EALDH1A1KDM1A
SCHEMBL8893944 0.62 KMT2A (0.46) NPY5RKDM4EALDH1A1MEN1KMT2A
Hydrochloric Acid SCHEMBL8905468 0.62 KMT2A (0.45) NPY5RKDM4EALDH1A1MEN1KMT2A
SCHEMBL8893955 0.61 NPY5R (0.40) KDRNPY5RALKEGFRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997020822-A1 QUINAZOLIN-2,4-DIAZIRINES AS NPY RECEPTOR ANTAGONIST NOVARTIS AG (CH) 1997-06-12 WO claimed