SCHEMBL8893944

SCHEMBL8893944

COCC(=O)NCc1ccc(Nc2nc(Nc3ccc(Cl)cc3)c3cccc(OC)c3n2)cc1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.46
CTNNB1 P35222 1/20 0.45
TCF7L2 Q9NQB0 1/20 0.45
TRPA1 O75762 1/20 0.43
CCNT1 O60563 1/20 0.42
CCNE1 P24864 1/20 0.42
CDK2 P24941 1/20 0.42
CDK9 P50750 1/20 0.42
ALDH1A1 P00352 2/20 0.42
MEN1 O00255 2/20 0.41
THRB P10828 1/20 0.41
NPY5R Q15761 2/20 0.41
POLB P06746 1/20 0.41
KDM4E B2RXH2 1/20 0.40
PKM P14618 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8905468 0.99 KMT2A (0.45) KMT2ACTNNB1TCF7L2TRPA1CCNT1
SCHEMBL8889844 0.93 NPY5R (0.48) CCNT1CCNE1CDK2CDK9NPY5R
SCHEMBL8893955 0.82 NPY5R (0.40) KMT2ACTNNB1TCF7L2CCNT1CCNE1
SCHEMBL8891133 0.81 NPY5R (0.46) CTNNB1TCF7L2TRPA1NPY5R
SCHEMBL8900365 0.81 SLC2A1 (0.49) KMT2AALDH1A1MEN1NPY5RKDM4E
SCHEMBL8890323 0.78 NPY5R (0.45) NPY5R
Hydrochloric Acid SCHEMBL8890553 0.77 NPY5R (0.44) NPY5R
SCHEMBL8898845 0.76 NPY5R (0.41) KMT2AALDH1A1MEN1NPY5RPOLB
SCHEMBL8901142 0.76 NPY5R (0.51) NPY5R
Hydrochloric Acid SCHEMBL8905477 0.75 NPY5R (0.40) KMT2AALDH1A1MEN1NPY5RPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997020822-A1 QUINAZOLIN-2,4-DIAZIRINES AS NPY RECEPTOR ANTAGONIST NOVARTIS AG (CH) 1997-06-12 WO claimed