SCHEMBL8890945

SCHEMBL8890945

Cc1ccc(Nc2nc(Nc3ccccc3)c3ccccc3n2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 9/20 1.00
PGK1 P00558 1/20 0.69
SLC2A1 P11166 1/20 0.68
MAPT P10636 3/20 0.67
LMNA P02545 2/20 0.67
TP53 P04637 1/20 0.67
ABCG2 Q9UNQ0 1/20 0.67
PTGS2 P35354 1/20 0.62
AURKA O14965 1/20 0.61
SRC P12931 1/20 0.61
GSK3B P49841 1/20 0.61
KDM4E B2RXH2 2/20 0.60
ALDH1A1 P00352 2/20 0.60
RXFP1 Q9HBX9 1/20 0.60
MAPK1 P28482 2/20 0.60
HTT P42858 2/20 0.60
KMT2A Q03164 2/20 0.60
XBP1 P17861 1/20 0.60
SMN1; SMN2 Q16637 1/20 0.60
GPR55 Q9Y2T6 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8900357 0.98 NPY5R (0.97) NPY5RPGK1SLC2A1MAPTLMNA
SCHEMBL2590203 0.98 NPY5R (0.97) NPY5RPGK1SLC2A1MAPTLMNA
SCHEMBL2591063 0.90 NPY5R (1.00) NPY5RSLC2A1TP53ABCG2AURKA
Hydrochloric Acid SCHEMBL6039677 0.89 NPY5R (0.96) NPY5RSLC2A1MAPTTP53ABCG2
SCHEMBL2592190 0.88 NPY5R (0.78) NPY5RPGK1SLC2A1MAPTLMNA
SCHEMBL8901062 0.86 NPY5R (0.84) NPY5RSLC2A1LMNAABCG2ALDH1A1
SCHEMBL8898077 0.86 NPY5R (0.84) NPY5RSLC2A1MAPTABCG2KDM4E
Hydrochloric Acid SCHEMBL8898758 0.84 NPY5R (0.81) NPY5RSLC2A1MAPTABCG2KDM4E
SCHEMBL8890555 0.84 NPY5R (1.00) NPY5RSLC2A1MAPTTP53ABCG2
Hydrochloric Acid SCHEMBL8900034 0.84 NPY5R (0.81) NPY5RSLC2A1LMNATP53ABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997020822-A1 QUINAZOLIN-2,4-DIAZIRINES AS NPY RECEPTOR ANTAGONIST NOVARTIS AG (CH) 1997-06-12 WO claimed